Target Details
| UniProt AC | T1QYY3 |
|---|---|
| Gene Symbol | int |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 9
- Clinical molecules 0
- Avg pChEMBL 6.17
Top Co-occurrence Targets
- pol 9 shared
Active Molecules (9)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AOHAOGINVKWHLM
|
6.4 | IC50 | 2 | — | |
CAZFYBUUYWZTRA
|
6.3 | IC50 | 2 | — | |
LQTUWUPNINPQTG
|
6.2 | IC50 | 2 | — | |
LXPSWRHIYZOHTR
|
6.2 | IC50 | 2 | — | |
QRSZRABLONQUBE
|
6.1 | IC50 | 2 | — | |
WCIWRYQMQLNIMG
|
6.1 | IC50 | 2 | — | |
JEKLJKGXYFFOIW
|
6.1 | IC50 | 2 | — | |
PZWIJHWZZUHCAR
|
6.0 | IC50 | 2 | — | |
LLUSSJQGFFRYIN
|
6.0 | IC50 | 2 | — |