Target Details
| UniProt AC | Q9YQ12 |
|---|---|
| Gene Symbol | protease |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00077 (RVP) |
Summary
- Multi-target molecules 178
- Clinical molecules 0
- Avg pChEMBL 8.87
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VEJOBLYVGLPABL
|
7.4 | Ki | 2 | — | |
JBHCPNAOYVCBLC
|
7.4 | Ki | 2 | — | |
FAXGPCHRFPCXOO
|
7.3 | Ki | 14 | — | |
MNHOXZBSLMSIDR
|
7.3 | IC50 | 2 | — | |
CWMBLJUBLZGJFU
|
7.2 | Ki | 2 | — | |
UPYUBPUDWRHOBW
|
7.1 | IC50 | 3 | — | |
UXOWGYHJODZGMF
|
7.1 | Ki | 2 | — | |
OSKMOKTVGGXEKD
|
7.1 | IC50 | 2 | — | |
PQJCVHDSBMYBNP
|
7.1 | Ki | 2 | — | |
RTQWXKCFXHCIFO
|
7.1 | Ki | 3 | — | |
JKHQJAXRLPWNHI
|
6.9 | Ki | 2 | — | |
XESKRTWBOYRKRZ
|
6.9 | Ki | 2 | — | |
TZHVWGUJONDDOT
|
6.8 | IC50 | 2 | — | |
RWJPHGJNZTXMGR
|
6.8 | IC50 | 3 | — | |
WKYBEGDEGRCZNF
|
6.6 | Kd | 3 | — | |
RXXJTASWFDWOMQ
|
6.6 | IC50 | 2 | — | |
GQKWNYLKLDCKEF
|
6.5 | Ki | 2 | — | |
YTBBVCQPJXFQBH
|
6.5 | Ki | 3 | — | |
LZJOGRNDENREKS
|
6.4 | IC50 | 2 | — | |
AAROLUGLGDXGEZ
|
6.4 | Ki | 2 | — | |
FZINVUNMMCVSEY
|
6.3 | IC50 | 2 | — | |
ZZGMOZUZSAJAML
|
6.3 | IC50 | 2 | — | |
SVOHWMZXBFVEHY
|
6.2 | Ki | 3 | — | |
XTNGUQKDFGDXSJ
|
6.2 | Ki | 3 | — | |
RWBIVIUXFGDQLF
|
6.2 | Ki | 2 | — | |
PZCSYTKHAKPNOQ
|
6.2 | Ki | 2 | — | |
BMXYVKCLBAGXOY
|
6.0 | Ki | 2 | — | |
YOBNNQXGIZIFRK
|
6.0 | IC50 | 2 | — |