Target Details
| UniProt AC | Q9Y6R4 |
|---|---|
| Gene Symbol | MAP3K4 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF19431 (MEKK4_N) PF00069 (Pkinase) |
Summary
- Multi-target molecules 7
- Clinical molecules 5
- Avg pChEMBL 6.89
KEGG Pathways (2)
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
7.5 | Kd | 1075 | — | |
JWNPDZNEKVCWMY
|
7.4 | Kd | 57 | Yes | |
VAARYSWULJUGST
|
7.2 | Kd | 119 | Yes | |
UBPYILGKFZZVDX
|
7.0 | Kd | 130 | Yes | |
WVUNYSQLFKLYNI
|
6.5 | Kd | 46 | Yes | |
ZBNZXTGUTAYRHI
|
6.5 | Kd | 102 | Yes | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — |