Target Details
UniProt ACQ9Y6M4
Gene SymbolCSNK1G3
Protein NameCasein kinase I isoform gamma-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF12605 (CK1gamma_C) PF00069 (Pkinase)
Summary
  • Multi-target molecules 112
  • Clinical molecules 4
  • Avg pChEMBL 6.82
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (112)
InChIKey pChEMBL Type Targets Clinical
GPKQGYSDQQIJLW 6.9 Ki 19
NEWAULHLLUCDPD 6.9 Ki 27
VWCSZVWZRTZNCH 6.8 Kd 8
CHTMRWQLNNRRFJ 6.8 Ki 70
DKXHSOUZPMHNIZ 6.8 Ki 51 Yes
GCBJDOWIQHMCMR 6.8 Ki 84
ISEDKXOMRIKZPK 6.8 Ki 13
LCKDESRGCHSHHO 6.8 Ki 18
MIKAKZKNMYZLDX 6.8 Ki 42
WINHZLLDWRZWRT 6.6 Kd 201 Yes
ASNQMAVHHGGQRB 6.6 Ki 14
LYNBNVBMAGDJRW 6.6 Ki 81
MGNQNQOSSLCUFP 6.6 Ki 12
NJPWCTYVEJIQBM 6.6 Ki 72
XPHWIERLJBFPFV 6.6 Ki 69
BGVLELSCIHASRV 6.5 Kd 12
BGVLELSCIHASRV 6.5 Kd 12
RJTQBPCQZQSZFF 6.5 Kd 9
LRESELHEXSUQGE 6.5 Ki 10
OWDRQHVEJIYVOI 6.5 Ki 47
YMIJUBCSOKSFRU 6.4 Ki 87
DKZYXHCYPUVGAF 6.4 Kd 112
YPTMZNNBDPEMOK 6.3 IC50 6
BPNUQXPIQBZCMR 6.3 Ki 60
GQHMZZXJWGPHDA 6.3 Ki 20
IMHKMKWSWHFKTM 6.3 Ki 13
IQNOGQGSOHNMCL 6.3 Ki 14
OMKZJNFKGWJFNX 6.3 Ki 8
VXYDJXMHISGSDA 6.3 Ki 59
WINHZLLDWRZWRT 6.3 Ki 66
XSDJOIOVIMPMHD 6.3 Ki 44
ZRQXCQXWTLVASO 6.3 Ki 36
CTNPALGJUAXMMC 6.2 Kd 151
FUMCKNCUEAQHCV 6.2 Ki 103
HWGZXYUOXGVACR 6.2 Ki 6
PYDWRLNPMMKKCI 6.2 Ki 7
XCHWBXBDZRJVDP 6.2 Ki 51
ZPVLRSVLOWVDJC 6.2 Ki 14
LFAHWMOZPVCJAY 6.2 Kd 8
JTVBXQAYBIJXRP 6.1 Kd 20
CALAEFSQWBJMDU 6.1 Ki 21
GEGCXGMFUYJULA 6.1 Ki 30 Yes
KIXUMWAIYCKDQQ 6.1 IC50 2
QYGMZFLXMWJYRJ 6.1 Ki 14
SPOBBSBKXJKGBG 6.1 Ki 16
XQVVPGYIWAGRNI 6.1 Ki 19
XYZNKCSDQRKAFR 6.1 Ki 53
DVVVOLSRHWJCHV 6.1 IC50 2
IXRCZLGBPPMVSP 6.1 Kd 9
BPNUQXPIQBZCMR 6.0 Kd 83 Yes
2D structure