Target Details
| UniProt AC | Q9Y6M4 |
|---|---|
| Gene Symbol | CSNK1G3 |
| Protein Name | Casein kinase I isoform gamma-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12605 (CK1gamma_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 112
- Clinical molecules 4
- Avg pChEMBL 6.82
KEGG Pathways (1)
Active Molecules (112)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DCDZHPAPVHOEDE
|
8.6 | IC50 | 3 | — | |
HQMKZJLJBDXPIZ
|
8.2 | IC50 | 3 | — | |
ZOFPTOHAYCZFGK
|
8.2 | IC50 | 3 | — | |
JNLRFODVNRITQL
|
8.1 | IC50 | 3 | — | |
UDFDIIVNIYWXDM
|
8.1 | Ki | 74 | — | |
RKUKAACYUCUJEE
|
8.0 | Ki | 58 | — | |
SYOXQXNUFXRNKH
|
8.0 | IC50 | 3 | — | |
FNUUVPCZCHTPPR
|
7.8 | IC50 | 3 | — | |
AAANQOJVZBRGRH
|
7.8 | IC50 | 3 | — | |
VAMRGLQMNCSXDM
|
7.7 | IC50 | 3 | — | |
SBFPHSVZEXSHTL
|
7.7 | Ki | 62 | — | |
XFWUTMHVDGPWLH
|
7.7 | Ki | 75 | — | |
WWXQFSIZULKTBJ
|
7.7 | IC50 | 3 | — | |
XCLVEFQLWKDCDX
|
7.6 | IC50 | 3 | — | |
WPBKIQLDOLQVHG
|
7.6 | IC50 | 3 | — | |
LBCTWIUPHHIYNO
|
7.6 | IC50 | 3 | — | |
XZTZFGIZKXWMMU
|
7.6 | IC50 | 3 | — | |
RBSCAZUMOUDJAV
|
7.5 | IC50 | 3 | — | |
UASMATGCQULMCR
|
7.5 | IC50 | 3 | — | |
CLEGDJQQHUTCOW
|
7.5 | Ki | 43 | — | |
LAFYDKMPJZTXHE
|
7.5 | IC50 | 3 | — | |
QAJPIJHWTGPUNZ
|
7.5 | Ki | 37 | — | |
QKBJAJHKKNYIJA
|
7.5 | IC50 | 3 | — | |
CQDQSVXDMSYUGR
|
7.5 | IC50 | 3 | — | |
HVEXJKQESNIDLM
|
7.4 | Kd | 10 | — | |
IWCAAHBDNLJZOI
|
7.4 | IC50 | 3 | — | |
KOHNRDPXFDZZJF
|
7.4 | Ki | 31 | — | |
VQGZDVVEVGGEKT
|
7.4 | IC50 | 3 | — | |
ADMFLILDQJSEIK
|
7.3 | Ki | 72 | — | |
KDFAUZONCVHIQC
|
7.3 | IC50 | 3 | — | |
RXZQIBZFLBEIRW
|
7.3 | IC50 | 3 | — | |
HBKRAHRIWQMIJU
|
7.2 | IC50 | 3 | — | |
PFYGLKQLEHKJBE
|
7.2 | IC50 | 3 | — | |
HPFYFRCFVGMDDC
|
7.2 | IC50 | 3 | — | |
VEPRLRDIGFBHAG
|
7.2 | IC50 | 3 | — | |
FUFJXSOSTJWEBE
|
7.2 | IC50 | 3 | — | |
AHTHSKQPKKMYPX
|
7.1 | IC50 | 3 | — | |
DBHMJFHKKRRBAC
|
7.1 | IC50 | 3 | — | |
JJJSCYSPSKBQAX
|
7.1 | Ki | 34 | — | |
UMTWTCVTRDYHQQ
|
7.1 | Ki | 56 | — | |
XBAIEEJJCJHBDL
|
7.1 | Ki | 17 | — | |
ZGZVRPRSFXRGCF
|
7.1 | Ki | 76 | — | |
ODPGGGTTYSGTGO
|
7.0 | Kd | 153 | — | |
XDJCLCLBSGGNKS
|
7.0 | Kd | 21 | — | |
BGVLELSCIHASRV
|
7.0 | Kd | 11 | — | |
LXVBELDBJGYFEM
|
7.0 | Ki | 20 | — | |
UTFXYGYVDDLJER
|
7.0 | Ki | 36 | — | |
YWTBGJGMTBHQTM
|
7.0 | Ki | 65 | — | |
BGYLKQWHNHTXJA
|
7.0 | IC50 | 3 | — | |
QSOOWYJFQWRIAY
|
6.9 | IC50 | 3 | — |