Target Details
| UniProt AC | Q9Y6K1 |
|---|---|
| Gene Symbol | DNMT3A |
| Protein Name | DNA (cytosine-5)-methyltransferase 3A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17980 (ADD_DNMT3) PF00145 (DNA_methylase) PF22855 (DNM3A_N) PF21255 (DNMT3_ADD_GATA1-like) PF00855 (PWWP) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 6.28
KEGG Pathways (4)
Associated Diseases (6)
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VMMRDFLDWHFNOX
|
7.0 | IC50 | 4 | — | |
LVKWYVRJCVWPCV
|
6.5 | IC50 | 4 | — | |
TXWSATBBJRPVTL
|
6.5 | IC50 | 5 | — | |
FAZNWIGAOYXZGW
|
6.4 | IC50 | 2 | — | |
FCEWTMLZJKEGGF
|
6.3 | IC50 | 3 | — | |
XDWLPZNQFCXPOO
|
6.2 | IC50 | 2 | — | |
JIMLOXBHGGUDPE
|
6.2 | IC50 | 4 | — | |
ZADSZMCBHZSPAY
|
6.1 | IC50 | 2 | — | |
QSYLKMKIVWJAAK
|
6.0 | IC50 | 2 | — | |
YOQISUXQHUFCLO
|
6.0 | IC50 | 3 | — | |
OCVYWWSLZGQEHY
|
6.0 | IC50 | 2 | — | |
VBJGTPSNFOGRFY
|
6.0 | IC50 | 2 | — |