Target Details
| UniProt AC | Q9Y6F1 |
|---|---|
| Gene Symbol | PARP3 |
| Protein Name | Protein mono-ADP-ribosyltransferase PARP3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) |
Summary
- Multi-target molecules 41
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (2)
Active Molecules (41)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XSPSNGRGTPWRHB
|
9.3 | IC50 | 3 | — | |
STSCRAGBCYODMY
|
9.0 | IC50 | 8 | — | |
BFJMBXAFUUTYIR
|
8.0 | Kd | 2 | — | |
MWIUPFYRAAIUMB
|
7.7 | IC50 | 3 | — | |
AUSDJKWCUGOMRT
|
7.7 | Kd | 2 | — | |
FCXORJBFYRYCGS
|
7.7 | Kd | 2 | — | |
IZPURWNXWPTMHH
|
7.7 | Kd | 2 | — | |
OKZVWHVKFPRNLX
|
7.7 | Kd | 2 | — | |
OOMGICXJISMCLR
|
7.7 | Kd | 2 | — | |
VYUKSMNSIRGBBM
|
7.7 | Kd | 2 | — | |
HWGQMRYQVZSGDQ
|
7.6 | Kd | 7 | — | |
GSHBUCNCWYHWKA
|
7.5 | Kd | 2 | — | |
KYPCNLJQBLPDKY
|
7.5 | Kd | 2 | — | |
LIGDLZRFUNWVFK
|
7.4 | Kd | 2 | — | |
ZDDPBFWHZOJFHF
|
7.3 | IC50 | 6 | — | |
AOLFJVDCFAXDOZ
|
7.3 | IC50 | 4 | — | |
FPMIUVGZAHMUQO
|
7.3 | Kd | 2 | — | |
BWTOWBOMDHKCDB
|
7.3 | IC50 | 7 | — | |
WKXCQZQWHUTWSY
|
7.3 | IC50 | 5 | — | |
FDLYAMZZIXQODN
|
7.3 | IC50 | 11 | — | |
HWGQMRYQVZSGDQ
|
7.2 | IC50 | 6 | — | |
LWIZMEPNSZKHGD
|
7.2 | IC50 | 3 | — | |
QNQFPYADHVFRKQ
|
7.2 | IC50 | 5 | — | |
GFHLWWHOLUWZLZ
|
7.2 | IC50 | 4 | — | |
HGEPGGJUGUMFHT
|
7.2 | Kd | 2 | — | |
NALBIBKGPRRCCO
|
7.2 | Kd | 2 | — | |
POAFYPSDLXGQBX
|
7.0 | Kd | 3 | — | |
MPXAEYSGFKRDQM
|
7.0 | IC50 | 7 | — | |
DENYZIUJOTUUNY
|
7.0 | IC50 | 5 | — | |
MHQFEYXRRZRKBA
|
6.9 | IC50 | 3 | — | |
UFCYAFSJOZTJKT
|
6.7 | IC50 | 3 | — | |
GGJVOTFHPYZESL
|
6.7 | IC50 | 4 | — | |
JNAHVYVRKWKWKQ
|
6.6 | Kd | 4 | — | |
PQXUCBRUEQVEIZ
|
6.6 | Kd | 3 | — | |
PCHKPVIQAHNQLW
|
6.5 | IC50 | 8 | — | |
HMABYWSNWIZPAG
|
6.5 | IC50 | 12 | — | |
HTRPLWGQNMXGRD
|
6.2 | IC50 | 3 | — | |
UYJZZVDLGDDTCL
|
6.2 | Kd | 8 | — | |
PZDZBZWWQUDTKX
|
6.1 | IC50 | 3 | — | |
KLGQSVMIPOVQAX
|
6.1 | IC50 | 7 | — | |
CHUANYXVPMSWFM
|
6.0 | IC50 | 3 | — |