Target Details
| UniProt AC | Q9Y618 |
|---|---|
| Gene Symbol | NCOR2 |
| Protein Name | Nuclear receptor corepressor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15784 (GPS2_interact) PF00249 (Myb_DNA-binding) |
Summary
- Multi-target molecules 423
- Clinical molecules 20
- Avg pChEMBL 7.34
KEGG Pathways (2)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WXWAPGNHECFJAW
|
6.5 | IC50 | 4 | — | |
SCZTZKHHRWDIJY
|
6.5 | IC50 | 2 | — | |
UDCHKWFFUPZXLN
|
6.5 | IC50 | 2 | — | |
QAJFPPXXVZWNQN
|
6.5 | IC50 | 3 | — | |
PFADLOXEKLDOIQ
|
6.4 | IC50 | 6 | — | |
ROCSVJSPJGRGIX
|
6.4 | IC50 | 4 | — | |
ATAYIUXFFSKHFW
|
6.4 | IC50 | 2 | — | |
UILCCVKVTDINGS
|
6.4 | IC50 | 3 | — | |
KYHKYEUYJZTRCP
|
6.4 | IC50 | 2 | — | |
MMKIXMJBZVVFRQ
|
6.4 | IC50 | 6 | — | |
RMNSKKUFRXPOEG
|
6.4 | IC50 | 2 | — | |
SNLPPFAZSJSJSF
|
6.4 | IC50 | 3 | — | |
PBGPTBJLOKADHP
|
6.3 | Kd | 2 | — | |
WFNAWUGSMGCUGF
|
6.3 | IC50 | 8 | — | |
HNNSHRLHFRPHCC
|
6.3 | IC50 | 4 | — | |
VJFKSXHAFLCLLP
|
6.3 | IC50 | 2 | — | |
NUUAPTZQDCCEPP
|
6.3 | IC50 | 2 | — | |
TUQZMESLDYEUSM
|
6.3 | IC50 | 2 | — | |
ANMZNMDSWZJYNP
|
6.3 | IC50 | 6 | — | |
BLVQHYHDYFTPDV
|
6.3 | Ki | 4 | — | |
CNAQOPITLAIDTC
|
6.3 | IC50 | 2 | — | |
GMTQIBOGHFJELF
|
6.3 | IC50 | 3 | — | |
OVOYFFMFJBJCRU
|
6.3 | IC50 | 5 | — | |
SRCGSXKCMDYLRX
|
6.3 | IC50 | 4 | — | |
NWDGFYIDKSNNQH
|
6.3 | IC50 | 8 | — | |
PZFYWPRLDKIIHM
|
6.3 | IC50 | 4 | — | |
BBHHBNFCYBGQHQ
|
6.3 | IC50 | 4 | — | |
NUNBOGCRDXXYGD
|
6.3 | IC50 | 2 | — | |
DVHSVOTUIFPGKP
|
6.2 | IC50 | 3 | — | |
IPJBYSCSCXDDEE
|
6.2 | IC50 | 3 | — | |
JFVYUMCLAOMZHX
|
6.2 | IC50 | 3 | — | |
JRYSTMMUZUGAAW
|
6.2 | IC50 | 4 | — | |
SIRNCVDOMIOFAK
|
6.2 | IC50 | 12 | — | |
YEJPAUXCGZXHNF
|
6.2 | IC50 | 3 | — | |
BGCPLWWYPZAURQ
|
6.2 | IC50 | 2 | — | |
DTUYIDRKQUOHOD
|
6.2 | IC50 | 3 | — | |
PSDULCGBSAPYKD
|
6.2 | IC50 | 2 | — | |
SMLFVHZWGKWRSD
|
6.2 | IC50 | 3 | — | |
BLVLSEPOIOLKDB
|
6.2 | IC50 | 13 | Yes | |
JOEWBFMDFCFWJV
|
6.2 | IC50 | 4 | — | |
LYCCCRFBRDLGGA
|
6.2 | IC50 | 6 | — | |
BBOZKUDSOWBNPX
|
6.2 | IC50 | 2 | — | |
DCHJMXBGNPORHN
|
6.2 | IC50 | 12 | — | |
OONGOCHJMMTGRJ
|
6.2 | IC50 | 12 | — | |
XIBYSMPUNMZEDF
|
6.2 | IC50 | 3 | — | |
FZTMVYQHIOEHIG
|
6.2 | IC50 | 4 | — | |
BYQQNBDKRJXLHR
|
6.1 | IC50 | 3 | — | |
ODMBSJLKYGMCQA
|
6.1 | IC50 | 2 | — | |
WNDZFLFSVTWZRB
|
6.1 | IC50 | 5 | — | |
YXJPLEKIYDOIFE
|
6.1 | IC50 | 4 | — |