Target Details
| UniProt AC | Q9Y618 |
|---|---|
| Gene Symbol | NCOR2 |
| Protein Name | Nuclear receptor corepressor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15784 (GPS2_interact) PF00249 (Myb_DNA-binding) |
Summary
- Multi-target molecules 423
- Clinical molecules 20
- Avg pChEMBL 7.34
KEGG Pathways (2)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHKLSMMMMRFDLK
|
7.1 | IC50 | 3 | — | |
NHIVVTDJMQAKAA
|
7.1 | IC50 | 2 | — | |
RJFQGJRGMDZGTD
|
7.1 | IC50 | 12 | — | |
CNDVZDSPNMUYDC
|
7.1 | Kd | 2 | — | |
JZZQCWSGCPALEP
|
7.1 | IC50 | 4 | — | |
MZVLQECJCSSXJD
|
7.1 | IC50 | 5 | — | |
VJXBYUITQBTTQM
|
7.1 | IC50 | 5 | Yes | |
PKWHZXFHRVODQW
|
7.0 | Kd | 2 | — | |
QMGDCUHFYVMSBA
|
7.0 | IC50 | 8 | — | |
UHPVVZUVOPNTDE
|
7.0 | IC50 | 12 | — | |
BEFOBMGNAJJGSD
|
7.0 | IC50 | 3 | — | |
PJXHIWAHCJGLOV
|
7.0 | Kd | 2 | — | |
CRNDOQUVHYQTBI
|
7.0 | Kd | 2 | — | |
FNEMPWZNAOCUEQ
|
7.0 | IC50 | 4 | — | |
LOEFBHPFPGYXOH
|
7.0 | IC50 | 4 | — | |
OEBYRDHGFUDTDM
|
7.0 | IC50 | 4 | — | |
UWJMLPAEGOKDNK
|
7.0 | IC50 | 12 | — | |
JTJKITJOSCGZOP
|
7.0 | IC50 | 2 | — | |
LHPSCRKAXVEHHI
|
7.0 | Kd | 2 | — | |
TWIPDOQQXDCJOF
|
7.0 | IC50 | 6 | — | |
VGUURLUFIOIIBI
|
7.0 | IC50 | 12 | — | |
DAWMVKMNSDXVNL
|
7.0 | IC50 | 3 | — | |
FRPLQLNSYVGWHG
|
7.0 | Kd | 2 | — | |
GQHSZFIWJYNXMV
|
7.0 | Kd | 2 | — | |
OQXGDFSYMGTLHG
|
7.0 | IC50 | 7 | — | |
UODZPFZHXUXNPW
|
7.0 | IC50 | 7 | — | |
ULHBYWCDCNACMV
|
7.0 | Kd | 2 | — | |
IZNDXKIRFLMXIW
|
6.9 | IC50 | 8 | — | |
FYAWEPJUGYZQDE
|
6.9 | IC50 | 3 | — | |
PCQQFHBCWBFDEF
|
6.9 | IC50 | 5 | — | |
XFBZAGGLERWKQC
|
6.9 | IC50 | 2 | — | |
KLPIKEBAJICFPE
|
6.9 | IC50 | 12 | — | |
AAMHUKDMAMABLC
|
6.9 | IC50 | 12 | — | |
CMXYMOWDNOBGHN
|
6.9 | IC50 | 2 | — | |
CRJOTIVIHHXBSQ
|
6.9 | IC50 | 12 | — | |
IUQBJPLGIIVXFD
|
6.9 | IC50 | 5 | — | |
JFVYUMCLAOMZHX
|
6.9 | IC50 | 2 | — | |
NMCXQPBZVFQDAA
|
6.9 | IC50 | 2 | — | |
HPFNQVXPHMIRLD
|
6.9 | Kd | 2 | — | |
RUVFSSHGAAUXCC
|
6.9 | Kd | 2 | — | |
YALNUENQHAQXEA
|
6.9 | IC50 | 13 | Yes | |
VLVGUAGNSVBLEP
|
6.9 | IC50 | 2 | — | |
IKCHZDNFNSMGAW
|
6.8 | IC50 | 6 | — | |
NCVXXLOPDSGPAS
|
6.8 | Kd | 2 | — | |
RIIWGLKYAIUMGL
|
6.8 | IC50 | 12 | — | |
YWLNYZXFIAFWSF
|
6.8 | IC50 | 3 | — | |
FEANGDQVGBXDMV
|
6.8 | IC50 | 8 | — | |
MAUCONCHVWBMHK
|
6.8 | IC50 | 12 | — | |
SMBGAUXQNOXKIW
|
6.8 | IC50 | 2 | — | |
BEGKXXXIAVVHRO
|
6.8 | IC50 | 3 | — |