Target Details
| UniProt AC | Q9Y618 |
|---|---|
| Gene Symbol | NCOR2 |
| Protein Name | Nuclear receptor corepressor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15784 (GPS2_interact) PF00249 (Myb_DNA-binding) |
Summary
- Multi-target molecules 423
- Clinical molecules 20
- Avg pChEMBL 7.34
KEGG Pathways (2)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YPXXHURYIWPWFC
|
7.4 | IC50 | 3 | — | |
HRNLUBSXIHFDHP
|
7.3 | IC50 | 7 | Yes | |
WVAPBIZHYDNDKJ
|
7.3 | Kd | 2 | — | |
JYBYRHHEZONZJB
|
7.3 | IC50 | 4 | — | |
WAEXFXRVDQXREF
|
7.3 | IC50 | 20 | Yes | |
JTDYUFSDZATMKU
|
7.3 | IC50 | 13 | Yes | |
VEYVMZYCTFXASW
|
7.3 | Kd | 2 | — | |
ZWFAWLKMTVUZHD
|
7.3 | Kd | 2 | — | |
QGZYDVAGYRLSKP
|
7.3 | IC50 | 7 | — | |
RSMQIIFSOGKAHA
|
7.3 | IC50 | 5 | — | |
VLMYLGPYYNFPET
|
7.3 | IC50 | 5 | — | |
JSNKRNRGCDDSLD
|
7.3 | IC50 | 12 | — | |
RYUAYVJJTOJXBO
|
7.3 | IC50 | 6 | — | |
MNBGRERVWNCCTM
|
7.3 | IC50 | 3 | — | |
SRIRSXLHDKCIBH
|
7.3 | IC50 | 3 | — | |
VZGLMYCTCYVSQK
|
7.3 | IC50 | 2 | — | |
LOWZFLCPRNMALN
|
7.2 | Kd | 2 | — | |
ULQVOSFGFYDDOI
|
7.2 | IC50 | 3 | — | |
VYBKJKUFXIAVJM
|
7.2 | IC50 | 12 | — | |
NCQBGEPYHDJVHE
|
7.2 | Kd | 2 | — | |
DUSGJNWURDFHSJ
|
7.2 | Kd | 2 | — | |
OXRFZTKVNBHUJF
|
7.2 | IC50 | 3 | — | |
BVQCFCYPFJOOAV
|
7.2 | IC50 | 4 | — | |
CMFSOZAEQZHYJF
|
7.2 | IC50 | 3 | — | |
FMAYUVHWYXXHME
|
7.2 | IC50 | 5 | — | |
GMTQIBOGHFJELF
|
7.2 | IC50 | 4 | — | |
JADLTHLIKQJHTH
|
7.2 | IC50 | 2 | — | |
WRMLHFIPUNMIQC
|
7.2 | IC50 | 4 | — | |
GHCWLYKERZOPPW
|
7.2 | IC50 | 8 | — | |
HECBRMPKGMWNPZ
|
7.2 | IC50 | 12 | — | |
WTXFMLFPFKCMHO
|
7.2 | IC50 | 3 | — | |
RRJDFENBXIEAPD
|
7.2 | IC50 | 4 | — | |
RALPPESOHBXWNC
|
7.2 | IC50 | 3 | — | |
UPGCHGPZKCQKNK
|
7.2 | IC50 | 8 | — | |
IZJMRCTZDBCUHT
|
7.2 | IC50 | 2 | — | |
QMGDCUHFYVMSBA
|
7.2 | IC50 | 8 | — | |
GPIZQXBFYQDCHM
|
7.2 | IC50 | 12 | — | |
JHDKZFFAIZKUCU
|
7.2 | IC50 | 13 | Yes | |
XQXZIMLBLPDARP
|
7.2 | IC50 | 6 | — | |
ZAIULUYKQLVQFH
|
7.2 | IC50 | 3 | — | |
ZPFRKIBHYHVPPO
|
7.2 | IC50 | 12 | — | |
NZBHFBGHVBAHOW
|
7.2 | IC50 | 4 | — | |
SBNOWXXHMKPULR
|
7.1 | IC50 | 5 | — | |
SFICPVORFVXNPV
|
7.1 | IC50 | 6 | — | |
OBQXNVXJMUPSRH
|
7.1 | IC50 | 8 | — | |
ALHGXUGKLZHEOY
|
7.1 | Kd | 2 | — | |
HFDUFQFVUVYKCX
|
7.1 | IC50 | 6 | — | |
NSKNUBYLLYGFAI
|
7.1 | IC50 | 4 | — | |
INVTYAOGFAGBOE
|
7.1 | IC50 | 15 | Yes | |
MVBJZEXEUAHMFY
|
7.1 | IC50 | 4 | — |