Target Details
| UniProt AC | Q9Y618 |
|---|---|
| Gene Symbol | NCOR2 |
| Protein Name | Nuclear receptor corepressor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15784 (GPS2_interact) PF00249 (Myb_DNA-binding) |
Summary
- Multi-target molecules 423
- Clinical molecules 20
- Avg pChEMBL 7.34
KEGG Pathways (2)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DUSGJNWURDFHSJ
|
7.9 | Kd | 2 | — | |
NDXNRYJTYFEIAB
|
7.9 | IC50 | 2 | — | |
ZCZXFHBXRHZTID
|
7.9 | IC50 | 4 | — | |
LMAFSGDNHVBIHU
|
7.9 | IC50 | 14 | Yes | |
OVUUBMMQUPSVRE
|
7.9 | IC50 | 4 | — | |
QHHUXNDUTCMUPI
|
7.9 | IC50 | 4 | — | |
VAMVTPLUGOPXBG
|
7.9 | Kd | 2 | — | |
RTKIYFITIVXBLE
|
7.9 | IC50 | 17 | Yes | |
ZXOPHZQDWCEBMO
|
7.9 | IC50 | 2 | — | |
QKNOLJBQLJGNKI
|
7.9 | Ki | 8 | Yes | |
LGXWGGZWHGRIBP
|
7.9 | Kd | 2 | — | |
URAHKMFXCBPDOS
|
7.9 | Kd | 2 | — | |
OICURQWOFDGPNS
|
7.8 | IC50 | 8 | — | |
BMFJBTSGDSIZBF
|
7.8 | Kd | 2 | — | |
JWOGUUIOCYMBPV
|
7.8 | IC50 | 17 | Yes | |
BJZKQPOYFARQTQ
|
7.8 | Kd | 2 | — | |
CZTGBCYDMXHKOW
|
7.8 | IC50 | 2 | — | |
ICQCMPQEFWZGRJ
|
7.8 | IC50 | 4 | — | |
MFKWDGAIRDGDTG
|
7.8 | IC50 | 5 | — | |
UHLSPCYTRWSAEL
|
7.8 | Kd | 2 | — | |
VOPDXHFYDJAYNS
|
7.8 | IC50 | 3 | — | |
ZJQCSPLCJRVKSH
|
7.8 | IC50 | 3 | — | |
LMHHLDISEZZCMW
|
7.8 | IC50 | 4 | — | |
DDJFEVNAMKGVES
|
7.8 | IC50 | 5 | — | |
KKWSSPSMAXPDHE
|
7.8 | IC50 | 4 | — | |
QOEJRHVNEAVQSB
|
7.8 | IC50 | 4 | — | |
RCDISRRXFZPOQI
|
7.8 | Kd | 2 | — | |
VSHFAZBXGXHGQO
|
7.8 | IC50 | 13 | Yes | |
HFFOCGFIJMCQCW
|
7.7 | IC50 | 8 | — | |
OFVVEEGKXCCFDK
|
7.7 | IC50 | 5 | — | |
XFCDIVOWAPYSPP
|
7.7 | IC50 | 5 | — | |
AENKNAKODODQJV
|
7.7 | IC50 | 6 | — | |
CIGOMCAFKVJNOA
|
7.7 | IC50 | 5 | — | |
CMDHJYUFAKFOCL
|
7.7 | IC50 | 12 | — | |
GBIQEYYBFBGNOZ
|
7.7 | IC50 | 5 | — | |
KKWSSPSMAXPDHE
|
7.7 | IC50 | 4 | — | |
QBKLIARRJUTMTQ
|
7.7 | IC50 | 7 | — | |
MCRHRRIGPAVFNY
|
7.7 | IC50 | 2 | — | |
MUNWAZFRKGVMPQ
|
7.6 | IC50 | 4 | Yes | |
HFBCSHFRHHWQIW
|
7.6 | Kd | 2 | — | |
IDDXSQZUXBDLBA
|
7.6 | Kd | 2 | — | |
UPWACBOVNACRFH
|
7.6 | Kd | 2 | — | |
KGDRBYRBESIING
|
7.6 | Kd | 2 | — | |
OXEVGGGODZSGHA
|
7.6 | IC50 | 4 | — | |
RTLKDFQWSQARBW
|
7.6 | IC50 | 11 | — | |
BQGAVSCJXIZWNC
|
7.6 | IC50 | 4 | — | |
CSOPPLVKBKVKFI
|
7.6 | Kd | 2 | — | |
HHEYZHSUZVJWFR
|
7.6 | Kd | 2 | — | |
MBLMLNTUJWHBSJ
|
7.6 | Kd | 2 | — | |
OHRURASPPZQGQM
|
7.6 | IC50 | 14 | — |