Target Details
| UniProt AC | Q9Y618 |
|---|---|
| Gene Symbol | NCOR2 |
| Protein Name | Nuclear receptor corepressor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15784 (GPS2_interact) PF00249 (Myb_DNA-binding) |
Summary
- Multi-target molecules 423
- Clinical molecules 20
- Avg pChEMBL 7.34
KEGG Pathways (2)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SFTGPJZKXBQVEB
|
8.4 | Kd | 2 | — | |
VSGFAZMSYAWCRX
|
8.4 | Kd | 2 | — | |
BGOQTCCTQXNVFG
|
8.4 | Kd | 2 | — | |
YRRVLBINSXVLFM
|
8.4 | IC50 | 12 | — | |
PMPMWIHRIXQLDE
|
8.4 | Kd | 2 | — | |
OVPRWXARIKXWMC
|
8.4 | Kd | 2 | — | |
NSEFNIYZBRIBKB
|
8.3 | IC50 | 2 | — | |
PTZIPKBVSWCPSC
|
8.3 | Kd | 2 | — | |
ZPAHLBXHWVNFMV
|
8.3 | IC50 | 15 | — | |
QPHJHMOKVYIJGF
|
8.3 | IC50 | 6 | Yes | |
PAWIYAYFNXQGAP
|
8.3 | IC50 | 15 | — | |
BZYQCFUKLXJLGU
|
8.3 | IC50 | 5 | — | |
RQYNXNGSTYGHRK
|
8.3 | IC50 | 13 | — | |
HUWFWFGYLSDNMK
|
8.3 | IC50 | 4 | — | |
MEJLVLMAJJRLCR
|
8.3 | IC50 | 9 | Yes | |
MFQWEVWWKYZTOJ
|
8.3 | Kd | 2 | — | |
ULYVQURTWGHWFS
|
8.3 | IC50 | 5 | — | |
PLSOXLGFMFFJOA
|
8.2 | Kd | 2 | — | |
LGAFZGSECXDYIR
|
8.2 | Kd | 2 | — | |
ROZOBAUWRLENHV
|
8.2 | Kd | 2 | — | |
FYAWEPJUGYZQDE
|
8.2 | IC50 | 4 | — | |
GHXAGWZSAKFQHQ
|
8.2 | IC50 | 4 | — | |
MWAKEAASVJSTMA
|
8.2 | Kd | 2 | — | |
LLBWUNKGCADDKQ
|
8.2 | IC50 | 5 | — | |
SOUWDYWQNTVVMP
|
8.2 | IC50 | 7 | Yes | |
XXLPOYMHJXIFCW
|
8.2 | Kd | 2 | — | |
JWOGUUIOCYMBPV
|
8.2 | IC50 | 3 | — | |
NFSPQSDLXYVMOK
|
8.1 | Kd | 2 | — | |
YRIQBTBEZQCHRT
|
8.1 | Kd | 2 | — | |
KWYJMURUTYYRHS
|
8.1 | IC50 | 5 | — | |
VGJQCRDFIWDPMP
|
8.1 | Kd | 2 | — | |
MHZUZIALEUTHIU
|
8.1 | IC50 | 4 | — | |
PDJURBSVOZANDU
|
8.1 | IC50 | 6 | — | |
LYUHXLDJCYYUNT
|
8.1 | IC50 | 4 | — | |
XRHLECJNJSLFEN
|
8.1 | IC50 | 6 | — | |
SOQPPTRKIZLQFU
|
8.1 | IC50 | 4 | — | |
NKJANSUNVHHIIX
|
8.1 | IC50 | 4 | — | |
PANMZVOPZWWAGR
|
8.1 | IC50 | 12 | — | |
WCZYLKXWWUKEBA
|
8.1 | IC50 | 5 | — | |
UYJHFLMXMBPUNA
|
8.0 | Kd | 2 | — | |
ZGKVKLQBOOZORR
|
8.0 | IC50 | 4 | — | |
KFIPMJYXLUAZAW
|
8.0 | IC50 | 2 | — | |
DAGWCJGDWGPDPA
|
8.0 | IC50 | 8 | — | |
HIKRXEASUUGCMM
|
8.0 | IC50 | 4 | — | |
LLMWWARHOHTUED
|
8.0 | Kd | 2 | — | |
TWNWMDWWEMZXEH
|
8.0 | IC50 | 4 | — | |
JLTPFXJCUXAIDA
|
8.0 | Kd | 2 | — | |
KQIAPLSDGQOLIK
|
8.0 | Kd | 2 | — | |
GYAXGYBIYNGRAF
|
7.9 | Kd | 2 | — | |
KFARIDCZFMIHEZ
|
7.9 | Kd | 2 | — |