Target Details
| UniProt AC | Q9Y616 |
|---|---|
| Gene Symbol | IRAK3 |
| Protein Name | Interleukin-1 receptor-associated kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF00069 (Pkinase) |
Summary
- Multi-target molecules 39
- Clinical molecules 12
- Avg pChEMBL 6.96
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (39)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ACJQMCQTSXRKNU
|
8.4 | IC50 | 2 | — | |
FQBRQRVXPUQKLG
|
8.2 | IC50 | 4 | — | |
DJVYXMINSBMUHH
|
8.0 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
8.0 | Kd | 220 | — | |
MWKSRKSEWLRPBL
|
8.0 | Kd | 1075 | — | |
DKZYXHCYPUVGAF
|
7.9 | Kd | 112 | — | |
HKSZLNNOFSGOKW
|
7.9 | Kd | 408 | — | |
ZUODKONSNNHSAJ
|
7.9 | IC50 | 7 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
LCVIRAZGMYMNNT
|
7.6 | Kd | 20 | — | |
MHXGEROHKGDZGO
|
7.6 | Kd | 10 | — | |
WKDACQVEJIVHMZ
|
7.6 | Kd | 46 | — | |
FQBRQRVXPUQKLG
|
7.5 | IC50 | 10 | — | |
KTEIFNKAUNYNJU
|
7.5 | Kd | 114 | — | |
HWXVIOGONBBTBY
|
7.5 | Kd | 27 | — | |
DJVYXMINSBMUHH
|
7.3 | IC50 | 8 | — | |
DJVYXMINSBMUHH
|
7.3 | IC50 | 8 | — | |
ALKJNCZNEOTEMP
|
7.1 | Kd | 55 | — | |
JOOXLOJCABQBSG
|
6.9 | Kd | 139 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
KOZFSFOOLUUIGY
|
6.6 | Kd | 88 | Yes | |
VXBAJLGYBMTJCY
|
6.5 | Kd | 34 | Yes | |
CXQHYVUVSFXTMY
|
6.4 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.4 | Kd | 149 | — | |
JGEBLDKNWBUGRZ
|
6.3 | Kd | 20 | Yes | |
ZCCPLJOKGAACRT
|
6.2 | Kd | 599 | — | |
OYONTEXKYJZFHA
|
6.2 | Kd | 69 | Yes | |
UXXQOJXBIDBUAC
|
6.1 | Kd | 21 | Yes | |
SNCZIVUNTWOQAF
|
6.1 | IC50 | 4 | — | |
WJRRGYBTGDJBFX
|
6.1 | Kd | 16 | Yes | |
CUIHSIWYWATEQL
|
6.1 | Kd | 61 | Yes | |
IYHHRZBKXXKDDY
|
6.0 | IC50 | 6 | — | |
WINHZLLDWRZWRT
|
6.0 | Kd | 201 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes |