Target Details
| UniProt AC | Q9Y5Y9 |
|---|---|
| Gene Symbol | SCN10A |
| Protein Name | Sodium channel protein type 10 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) |
Summary
- Multi-target molecules 171
- Clinical molecules 0
- Avg pChEMBL 7.05
Associated Diseases (1)
Active Molecules (171)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXFWXFPSQUGQID
|
6.9 | IC50 | 2 | — | |
KUCYRCUGXDBLAO
|
6.9 | IC50 | 2 | — | |
MFMKNWRHVZVDBH
|
6.8 | IC50 | 2 | — | |
IKWWVCWYCSDROX
|
6.8 | IC50 | 2 | — | |
VYANEYBOMGSJQI
|
6.8 | IC50 | 2 | — | |
BDNWHXABGMGJIY
|
6.8 | IC50 | 2 | — | |
KHYNGGVKOMNOKG
|
6.7 | Ki | 2 | — | |
FCXMXLXAUSDGLN
|
6.7 | IC50 | 2 | — | |
IJZKTKBPFIPSJP
|
6.7 | IC50 | 2 | — | |
KDRVGEHIJOXPBO
|
6.7 | IC50 | 2 | — | |
CNJHIRPGEOQTTC
|
6.6 | IC50 | 2 | — | |
JWDYVXBLOYZJLX
|
6.6 | IC50 | 2 | — | |
XEDSOXUCOFSPMG
|
6.6 | IC50 | 2 | — | |
TTXHVPIJWCJKLK
|
6.6 | IC50 | 2 | — | |
YTHVKXJUOMIOFP
|
6.6 | IC50 | 3 | — | |
XBCPDKDJZGECMM
|
6.5 | IC50 | 2 | — | |
NFUBWILZNIMKMD
|
6.5 | IC50 | 2 | — | |
LNRALXGEGPHUEQ
|
6.5 | IC50 | 2 | — | |
LQBHOJPQVSFKSZ
|
6.5 | IC50 | 2 | — | |
OWKCSDFZMUWPDJ
|
6.5 | IC50 | 2 | — | |
BXOIJQLSRAKHJK
|
6.5 | IC50 | 2 | — | |
CGHVTPLFSBFCMC
|
6.5 | IC50 | 2 | — | |
CRIVLAVCQBIGSC
|
6.5 | IC50 | 2 | — | |
JYSHLENEZRKPDK
|
6.5 | IC50 | 2 | — | |
XUGUKAXHZIOGLG
|
6.5 | IC50 | 2 | — | |
OFVXFYHEMPXWQX
|
6.5 | IC50 | 2 | — | |
CCIDREHXLARDHU
|
6.4 | IC50 | 2 | — | |
ROVOFYSXQNIDPA
|
6.4 | IC50 | 2 | — | |
FJCCQQXMASEMDV
|
6.4 | IC50 | 2 | — | |
QCDCHYCAWONKAY
|
6.4 | IC50 | 2 | — | |
HPURRFIKNKVIFS
|
6.4 | IC50 | 2 | — | |
LXNIGQIGUFGETR
|
6.4 | IC50 | 2 | — | |
RTLVFTLHWCSMKT
|
6.4 | IC50 | 2 | — | |
PKVSOUFAHPBDDR
|
6.4 | IC50 | 2 | — | |
AMSKTYLOKZVQRX
|
6.3 | IC50 | 3 | — | |
NJGHOWOIRIXDKZ
|
6.3 | IC50 | 2 | — | |
QUPOUNZWMBLXGJ
|
6.3 | IC50 | 2 | — | |
IQNGIYJIIGTIOM
|
6.3 | IC50 | 2 | — | |
PJWLKPFEAXQJNQ
|
6.3 | IC50 | 2 | — | |
FCWGDENQRAUXMY
|
6.3 | IC50 | 2 | — | |
KICOFBPOACPQPG
|
6.3 | IC50 | 2 | — | |
MXMPAEFBKRMQFZ
|
6.3 | IC50 | 2 | — | |
QWVHTZXEQKODDC
|
6.3 | IC50 | 2 | — | |
XBAKWGXDYRBWJH
|
6.3 | IC50 | 2 | — | |
KYXKKYKXKUCVDJ
|
6.3 | IC50 | 2 | — | |
VEEQSZWXUOUXPZ
|
6.3 | IC50 | 5 | — | |
NUSVQLKNXPBOPF
|
6.3 | IC50 | 2 | — | |
DITZNZYXKSFLJE
|
6.2 | IC50 | 2 | — | |
BSCTXVDJXNZALB
|
6.2 | IC50 | 2 | — | |
MOVOFFZXYKIKPP
|
6.2 | IC50 | 2 | — |