Target Details
| UniProt AC | Q9Y5Y9 |
|---|---|
| Gene Symbol | SCN10A |
| Protein Name | Sodium channel protein type 10 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) |
Summary
- Multi-target molecules 171
- Clinical molecules 0
- Avg pChEMBL 7.05
Associated Diseases (1)
Active Molecules (171)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DMQWJYJEJRIDBI
|
7.4 | IC50 | 2 | — | |
BJWSTFAHQAKCBG
|
7.4 | IC50 | 2 | — | |
UXNUHKSSUVUOKZ
|
7.4 | IC50 | 2 | — | |
FPKSPIQOEJACSE
|
7.4 | IC50 | 2 | — | |
PIQAUSNVLROXMR
|
7.4 | IC50 | 2 | — | |
GGKJOYYMGVWXAT
|
7.3 | IC50 | 2 | — | |
IWRIRVFYRTUDIJ
|
7.3 | IC50 | 2 | — | |
BMYFAIFEOQGCTL
|
7.3 | IC50 | 2 | — | |
JLOCNBNTRGBNSU
|
7.3 | IC50 | 2 | — | |
IJLRJKVKJNUIJD
|
7.3 | IC50 | 2 | — | |
VWKUYSDQOUJGJG
|
7.3 | IC50 | 2 | — | |
AXDMEYZFXMOJQC
|
7.3 | IC50 | 2 | — | |
AKDINRARGVIZNO
|
7.3 | IC50 | 2 | — | |
URUKPZGNTWPRGW
|
7.3 | IC50 | 2 | — | |
WGGALQWPTKGQLX
|
7.3 | IC50 | 2 | — | |
YVUQSNJEYSNKRX
|
7.3 | IC50 | 36 | — | |
FAHBRZBMNSAQQB
|
7.2 | IC50 | 2 | — | |
FDMPUHDISMOMNB
|
7.2 | IC50 | 2 | — | |
HAHBFCDZJMZPDT
|
7.2 | IC50 | 2 | — | |
UFVVLUUDTNDRGT
|
7.2 | IC50 | 2 | — | |
IHQIUCIHAHGGQF
|
7.2 | IC50 | 2 | — | |
ZOFYFABDAAWNLG
|
7.2 | IC50 | 2 | — | |
GOXQSPDBNHQSLA
|
7.2 | IC50 | 2 | — | |
IHXQTRXZYHPGIQ
|
7.2 | IC50 | 2 | — | |
XMZFDPKNGIFRLZ
|
7.2 | IC50 | 2 | — | |
GFDFBVYVIAOKEU
|
7.2 | IC50 | 2 | — | |
CUVWAXHFLWGMGR
|
7.2 | IC50 | 2 | — | |
QDWZJQPXKINAHW
|
7.2 | IC50 | 2 | — | |
XQOGUSYHWGLZNJ
|
7.2 | IC50 | 2 | — | |
ICZIAJCVIIUREC
|
7.2 | IC50 | 2 | — | |
NDMNISGHBWDHTB
|
7.1 | IC50 | 2 | — | |
CKTPSKKTZVSXLI
|
7.1 | IC50 | 2 | — | |
QPACDKOMDYHWIR
|
7.1 | IC50 | 2 | — | |
FWASJBQVSBHBNK
|
7.1 | IC50 | 2 | — | |
AQMSMCUTJNXRFL
|
7.0 | IC50 | 2 | — | |
GHXUGFVKIDRBGU
|
7.0 | IC50 | 2 | — | |
ROWKGBJMLVUFFH
|
7.0 | IC50 | 2 | — | |
UMDJUPAXVBHNKS
|
7.0 | IC50 | 2 | — | |
IBHSESFTJVMJEA
|
7.0 | IC50 | 2 | — | |
MASHRDPYQKFCAR
|
7.0 | IC50 | 2 | — | |
JCPHCHCAKXVPLC
|
7.0 | IC50 | 2 | — | |
CBWXHMITTMOYOY
|
7.0 | IC50 | 2 | — | |
OVWZROCNURWRKK
|
7.0 | IC50 | 2 | — | |
PRDWHZNGVONJAX
|
7.0 | IC50 | 2 | — | |
UTKZKXRKSFATLD
|
7.0 | IC50 | 2 | — | |
CEWKJGUDXOKCAF
|
7.0 | IC50 | 2 | — | |
MFOFLSYIDKCECT
|
7.0 | IC50 | 2 | — | |
FKRJOLGOCURNRA
|
6.9 | IC50 | 2 | — | |
KYRYYQRTAJIXDA
|
6.9 | IC50 | 2 | — | |
ZXKIOHRLQVWVGA
|
6.9 | IC50 | 2 | — |