Target Details
| UniProt AC | Q9Y5Y9 |
|---|---|
| Gene Symbol | SCN10A |
| Protein Name | Sodium channel protein type 10 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) |
Summary
- Multi-target molecules 171
- Clinical molecules 0
- Avg pChEMBL 7.05
Associated Diseases (1)
Active Molecules (171)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CSKLRKQUNQCFCW
|
9.0 | IC50 | 2 | — | |
MDLXULGUOHLVMN
|
9.0 | IC50 | 2 | — | |
KFGUDEORIBZTGM
|
8.7 | IC50 | 2 | — | |
MLDMXXWILKZITA
|
8.7 | IC50 | 2 | — | |
ONXXBNABQCHJHC
|
8.7 | IC50 | 2 | — | |
OZJSEVZVZWZBIT
|
8.7 | IC50 | 2 | — | |
XNAAGHKLQDFJAV
|
8.5 | IC50 | 2 | — | |
OFJWZNKJBMVLPX
|
8.3 | IC50 | 2 | — | |
MEEMNCAUXAWBBT
|
8.2 | IC50 | 2 | — | |
CQIXHVVDGNOBRL
|
8.2 | IC50 | 2 | — | |
DSGSRMJPDQBTMM
|
8.2 | IC50 | 2 | — | |
DDGYZFJJKXLJOG
|
8.1 | IC50 | 2 | — | |
JJCBTWUQVASSGZ
|
8.0 | IC50 | 2 | — | |
OJGBGGHWKBSYTM
|
8.0 | IC50 | 2 | — | |
INIMUMMAVCNJFA
|
8.0 | IC50 | 2 | — | |
JKAMBBDGLZFTHQ
|
8.0 | IC50 | 2 | — | |
QYLLDXJQSXDYLQ
|
8.0 | IC50 | 2 | — | |
AJZDQSWVXBSGJM
|
7.9 | IC50 | 2 | — | |
KDVYWGKDSHINDP
|
7.9 | IC50 | 2 | — | |
IDCLDFZOZFUTLI
|
7.9 | IC50 | 2 | — | |
UHWLWOOUNBNZHS
|
7.9 | IC50 | 2 | — | |
IVBTXSATVJWRLA
|
7.8 | IC50 | 2 | — | |
UUAIQHMLXPMLDV
|
7.8 | IC50 | 2 | — | |
YXHMFJXQQXHKRO
|
7.8 | IC50 | 2 | — | |
OGNHUCWKIBGDPU
|
7.8 | IC50 | 2 | — | |
ZUFQSMFAKHTNSW
|
7.8 | IC50 | 2 | — | |
SXHSUVHECGYYMY
|
7.8 | IC50 | 2 | — | |
GOHNZFHVWZRGGX
|
7.7 | IC50 | 2 | — | |
DMUGWPYKKXFQFR
|
7.7 | IC50 | 2 | — | |
WLRVZQGFKCYIOQ
|
7.7 | IC50 | 2 | — | |
WSAJJTWYTKFRMU
|
7.7 | IC50 | 2 | — | |
OJJVDLJKYRQHKJ
|
7.7 | IC50 | 2 | — | |
JNNYSEIQBAVVNL
|
7.6 | IC50 | 2 | — | |
GFUFBVLEJPJQBR
|
7.6 | IC50 | 2 | — | |
GIJKDQHCVRCMIN
|
7.6 | IC50 | 2 | — | |
XLENMSSHHOXWHN
|
7.6 | IC50 | 2 | — | |
BVWMEUDWRCWKGL
|
7.5 | IC50 | 2 | — | |
XENPFDQDTNUZPA
|
7.5 | IC50 | 2 | — | |
FZRXMWNNMIDCAX
|
7.5 | IC50 | 2 | — | |
HJTNQQWICWEECK
|
7.5 | IC50 | 3 | — | |
POWGSPMXXFULOC
|
7.5 | IC50 | 2 | — | |
XFYJZSKHXSPHJR
|
7.5 | IC50 | 2 | — | |
XUEHBVFEQMVDHJ
|
7.5 | IC50 | 2 | — | |
IVXWSJDIJWTMBP
|
7.5 | IC50 | 2 | — | |
GCVAXVXEWOIGNP
|
7.5 | IC50 | 2 | — | |
OFZBNADUYSHVNR
|
7.5 | IC50 | 2 | — | |
UEAAJOBUYFZGHL
|
7.5 | IC50 | 2 | — | |
KWARURQEBURTJY
|
7.5 | IC50 | 2 | — | |
YWQDQDUGUYEIPV
|
7.4 | IC50 | 2 | — | |
ZRKHPQPMAITAEP
|
7.4 | IC50 | 2 | — |