Target Details
UniProt ACQ9Y5S2
Gene SymbolCDC42BPB
Protein NameSerine/threonine-protein kinase MRCK beta
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00130 (C1_1) PF00780 (CNH) PF08826 (DMPK_coil) PF15796 (KELK) PF25346 (PH_MRCK) PF00069 (Pkinase)
Summary
  • Multi-target molecules 202
  • Clinical molecules 5
  • Avg pChEMBL 8.43
Top Co-occurrence Targets
Active Molecules (202)
InChIKey pChEMBL Type Targets Clinical
RJTXALMLSLHCBH 7.7 Ki 3
NZNKOTVUZKHUSO 7.7 Ki 3
ZBDVDUIDYLZRJY 7.7 Ki 3
XFZYXYYYAMPVQK 7.7 Ki 2
GMYLSPYRJFWZRH 7.7 Ki 3
JTQOEKSUZBGXSZ 7.5 Ki 2
AOMUHYVRSKACNP 7.5 Ki 3
BLMKBLDBMAAGCC 7.5 Ki 3
HHGYNBXPZXZDBW 7.5 Ki 2
JTVBXQAYBIJXRP 7.5 Kd 20
FJHBZDZOSWVMSE 7.4 Ki 4
UZXCLKOZEMNTRB 7.4 Ki 3
JDIAOFCAAPMAGG 7.4 Ki 4
SCCMLQDEEDXQCZ 7.4 Ki 3
VHZNRUKXHPDXMR 7.4 Ki 4
RCADYZZSAWVHPR 7.4 Ki 4
HKSZLNNOFSGOKW 7.4 Kd 213
JWHQVVCSFIEMOB 7.4 Ki 3
LIZZRPJKAHJFGK 7.3 Ki 2
LNNCCLWHYORZTQ 7.3 Ki 3
KQDJZQWFJGSGBV 7.3 Ki 3
GJJMACISLUAOSI 7.3 Ki 3
XOMYQWBAFPYLRJ 7.3 Ki 3
IAUJYGJQLIMGNK 7.2 Ki 3
XETULWHBEZYEEP 7.2 Ki 3
FATRZQZLGUYQAN 7.2 Ki 3
IYUJRKGSEGCDSO 7.2 Ki 3
QUEIBWXZNMHZJD 7.1 Ki 4
AAKSFEZTNVXTKW 7.1 Ki 3
BPNUQXPIQBZCMR 7.0 Kd 83 Yes
HSUOPPIVYDGQEK 7.0 Ki 3
PBCZSGKMGDDXIJ 7.0 Kd 68 Yes
ASUGUQWIHMTFJL 6.9 Kd 18
OOPBTUDJGYIBIK 6.9 Ki 3
XPXCOKMZDASLDV 6.9 Ki 3
JWANSGWTSANRKI 6.9 Ki 2
FQNAKYCJWNZWHP 6.8 Ki 2
OOIZHXBHVKIGFO 6.8 Ki 3
XJSRTZCKTBCQLJ 6.7 Ki 3
OYZQKRFHAOKQNG 6.7 Ki 3
KHGJZRYHXCGFAZ 6.7 Ki 3
CXQHYVUVSFXTMY 6.5 Kd 154
SEJGTFPOEJWEGG 6.5 Kd 149
LMNVPKCUVZQIRI 6.5 Ki 2
MFGGOUDCVSWDFW 6.5 Ki 2
PRFFEESGSLBEAJ 6.5 Ki 3
VJHNKUNZCKSWRH 6.4 Ki 2
MCFSCRWDEDSWMA 6.2 Ki 3
ZCCPLJOKGAACRT 6.2 Kd 599
HHZIURLSWUIHRB 6.0 Kd 57 Yes
2D structure