Target Details
UniProt ACQ9Y5S2
Gene SymbolCDC42BPB
Protein NameSerine/threonine-protein kinase MRCK beta
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00130 (C1_1) PF00780 (CNH) PF08826 (DMPK_coil) PF15796 (KELK) PF25346 (PH_MRCK) PF00069 (Pkinase)
Summary
  • Multi-target molecules 202
  • Clinical molecules 5
  • Avg pChEMBL 8.43
Top Co-occurrence Targets
Active Molecules (202)
InChIKey pChEMBL Type Targets Clinical
QIOYFTZXBUZDSU 8.4 Ki 4
VTSLKIKDRBEGHX 8.4 Ki 3
LIZZRPJKAHJFGK 8.4 Ki 3
CGAGHKVPUASFJA 8.4 Ki 3
YDNXKPCILIWEGN 8.4 Ki 3
DVJSEIPSQLATHC 8.3 Ki 2
XULPQBFJASSWNQ 8.3 Ki 2
GBPXRWHRMNNALK 8.3 Ki 3
HKSZLNNOFSGOKW 8.3 IC50 408
SLDBVCHNZQQYKJ 8.3 Ki 3
BLMKBLDBMAAGCC 8.3 Ki 3
AZPUPQOGWVZSMS 8.2 Ki 2
KTDHNPKPSLZNRH 8.2 Ki 4
YEYOMHXUIKGONI 8.2 Ki 3
NVVLAIWWHAUHCF 8.2 Ki 4
TXPWZLKSGPRZAK 8.2 Ki 3
NFCAFNZSFOMNSD 8.2 Ki 3
NKMAMJNZKBGBFO 8.2 Ki 3
MRRXULDDEFCYAJ 8.2 Ki 3
XWQDAOOPQZIBIA 8.2 Ki 4
MUWPCRFJUPJCRM 8.1 Ki 4
NZNKOTVUZKHUSO 8.1 Ki 3
GRFYVFBPFKGUQO 8.1 Ki 2
HBYWJFGYPWTOHQ 8.1 Ki 3
DGPJCEDEJQDQFA 8.1 Ki 3
NXMNDVLAHWOSJG 8.1 Ki 3
XNAZVKJDUOIJBC 8.1 Ki 2
VKUWSTCDZXVNIT 8.1 Ki 4
MWKSRKSEWLRPBL 8.1 Kd 1075
FKFKNJHNUIUXHO 8.1 Ki 3
FNAPEKSJRDLQRC 8.0 Ki 4
HUXWDCVBFRJBIH 8.0 Ki 3
ULRKTUMEMQVQRV 8.0 Ki 3
SHMZVLGXEVPHCQ 8.0 Ki 4
XHAAAVYBPJTBLP 8.0 Ki 2
CGAGHKVPUASFJA 8.0 Ki 3
BTNHOAWDPXMJLS 7.9 Ki 2
LHCKGRAGUJSIPB 7.9 Ki 3
MQCSALLMDILSGX 7.9 Ki 3
IXBGOIVJRMXGGE 7.9 Ki 3
PUIKISPVMMUIMT 7.9 Ki 4
ZILLQAUSVGQYOB 7.9 Ki 4
VLFYWLXMVQEGMJ 7.9 Ki 3
OAWQMCAPBKNNRM 7.8 Ki 3
MRRXULDDEFCYAJ 7.8 Ki 3
VKORCHLUUJGKEE 7.8 Ki 3
IPEXHQGMTHOKQV 7.8 Kd 12
ADGQNANENRDMEA 7.8 Ki 4
DSQFKUKVDCXORL 7.8 Kd 4
DXZAHRFNIIHHLC 7.7 Ki 4
2D structure