Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
OJFKDXVECGWNTB 7.9 Ki 2
OLQOHRMMVIEWDK 7.9 Ki 2
WAIZFEIVFOBJJX 7.9 Ki 8
BOQXUEKBVIXPKQ 7.9 Ki 2
GMFZCHLJVCOHAA 7.9 Ki 2
NESASFDNMLPZIR 7.9 IC50 2
XEKHYAPKOUIALX 7.9 Ki 2
XOGNVWVGXPSTMU 7.9 Ki 2
BFGRVRCTCWRWNN 7.8 Ki 2
DGCHOADTPWCGNV 7.8 Ki 2
HGLGWLWXYRAXPK 7.8 Ki 2
JJHWOWWUTNJQFO 7.8 Ki 2
NWKCIVHGGAEYQL 7.8 Ki 2
QSADIYOOZUGQQY 7.8 Ki 4 Yes
CNAHRPLBYREXJE 7.8 Ki 2
FLZMPXADQFZKGE 7.8 Ki 2
LSLKPVQOFVGVSL 7.8 Ki 2
QJPBTFRGWJLPSI 7.8 Ki 2
UKKROAMTGBMPKN 7.8 Ki 2
CRMAPALWSALKCW 7.8 Ki 4
MVHBNHUOEFGIBK 7.8 Ki 2
QEAGVVCSVDNICD 7.8 Ki 2
RMQURPVWFQWESL 7.8 Ki 2
UNQMLUWBMWGIRY 7.8 Ki 4
ZNBGWUKXSAVPOB 7.8 Ki 2
CEQAEEYYVALJJW 7.8 Ki 4 Yes
GVCJWYDRTZSVBG 7.8 Ki 2
HAZUWABOLNYYCL 7.8 Ki 4 Yes
LJIRQKCQUPMGIY 7.8 Ki 3
QPCGSLWGRJGHNY 7.8 Ki 5
HFOWUCXCCMJFIB 7.7 Ki 2
OCBPATCVPDEFSN 7.7 Ki 2
GFCZIYIOXQZPFE 7.7 Ki 2
BOAJEIFQZOFOCK 7.7 Ki 2
BTEMXIHCAGOPHX 7.7 IC50 9
GILFIGFCCGSEPL 7.7 Ki 2
ISCCKNOQYHJXGM 7.7 Kd 2
KLOWQCMHDZVUBY 7.7 Ki 2
LIGSZPKQICJMNT 7.7 Ki 2
LKRTVYMJTLSROG 7.7 Ki 2
QPMSLQGYNLIUOH 7.7 Ki 2
UCIGGFFPBMFKPO 7.7 Kd 2
WMIWAHNZDCLEIJ 7.7 Ki 2
XSOYKCANSOSZRB 7.7 Ki 2
NESASFDNMLPZIR 7.7 Ki 2
HBSKTTXZUZBHRU 7.7 Ki 2
NCDVDCYFZPSORZ 7.7 Ki 2
KPJNSSGIUKWMPK 7.6 Ki 2
SBAQYPMYNRQKBF 7.6 Ki 3
SPBSCPKJFSEOAQ 7.6 Ki 2
2D structure