Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
DREYZGCIOLBBDK 8.1 IC50 2
LWZLGSJIXYLYMG 8.1 Ki 2
NZDANPPRKVYGPL 8.0 Ki 9
GHBUBJMRVNPMSE 8.0 Ki 2
KRWTTWQHPPVRDH 8.0 Ki 2
ZMOPTLXEYOVARP 8.0 Ki 14 Yes
CRTYYKOCTYXVIC 8.0 Ki 2
HKPCPMXAVHHCKQ 8.0 Ki 2
OHIPOORSUHEFRE 8.0 Ki 2
PMTYUERLXGUADP 8.0 Ki 2
JVYJGMIWWGWCJQ 8.0 Ki 4 Yes
KEILDXMRCDDBSQ 8.0 Ki 2
SSRXSLUJFGLVJI 8.0 Ki 2
VTPCFOYQLMVYRO 8.0 Ki 4 Yes
WWSHLNJFRHBFML 8.0 Ki 2
AQRDKFVOYVDLCT 8.0 Ki 2
BWTPAXCLYPICBF 8.0 Ki 2
DLEHGKOYLBSEGL 8.0 Ki 2
FZXKHRPYMDMOOX 8.0 Ki 2
IOCXEAYYBZJHHK 8.0 Ki 2
LGUCWRBFHWJFMF 8.0 Ki 2
QDMPFGBUXBHFTH 8.0 Ki 2
VTMJTHCQLMVWGT 8.0 Ki 4
XUIQQBLOOOYXMH 8.0 IC50 2
XYYGFCDTBHAUSN 8.0 Ki 4
KVVJWXBYIMMQTR 8.0 Ki 2
MJOSWDSZKHMYMF 8.0 Ki 2
XYYGFCDTBHAUSN 8.0 Ki 4 Yes
BDUVGZUKNGPFEZ 8.0 Ki 6
CPILYYRWNUVSHU 8.0 Ki 2
CQKVWEYZUVUWJT 8.0 Ki 2
DYUSEVKSEDICGM 8.0 Ki 6 Yes
GTLCRPKCYIDHGJ 8.0 Ki 4 Yes
KUYNMYBNRQCGCC 8.0 Ki 6 Yes
NQDGCGNKNJWZHP 8.0 Ki 5
NZPOPKFDIKJIRC 8.0 Ki 2
RAEJZLUTUUNZSA 8.0 Ki 2
XFSHNAXXKOSENG 7.9 IC50 2
BOQXUEKBVIXPKQ 7.9 IC50 2
CCXHRSBOCZSERO 7.9 Ki 2
FCAUWCISADYVAP 7.9 Ki 4
PRLJSGHDMGISHB 7.9 Ki 2
RSHJCGZZSGNBHO 7.9 Ki 2
KGHXTHFMZMFRTA 7.9 Ki 2
NTYJJOPFIAHURM 7.9 Ki 4
ALZTYVXVRZIERJ 7.9 Ki 2
BQBXKSFQNZVIMG 7.9 Ki 4 Yes
CQWSBUJEGUSBFA 7.9 Ki 2
HRDUUEDPDCVSJF 7.9 Ki 2
MFLUAACJGOHFDP 7.9 Ki 4 Yes
2D structure