Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
OICXGVDCXUDGKS 8.2 Ki 4 Yes
SURMDNBXOGRWFS 8.2 Ki 4 Yes
WNWALBVQAAIULR 8.2 Ki 2
YYOXBGHALUHPAP 8.2 IC50 2
DUKRHXPXPYNWKN 8.2 Ki 4 Yes
FNSGKKGXUCTTRV 8.2 Ki 4
YKCOYIKIANOWTN 8.2 Ki 6 Yes
FWJKAQILVAFVQQ 8.2 Ki 6 Yes
CIIDBUDXODMZQH 8.2 Ki 2
OVYKUTIVKUFDSG 8.2 Ki 2
WXQZQMBHXNYUDM 8.2 Ki 2
JJPGVZOMHHYPJU 8.2 Ki 2
HZNTWQAMIOKCMC 8.2 IC50 2
QKGFAFCTWJXMJH 8.2 Ki 2
SYZMKZBTICLWQD 8.2 Ki 2
DIMAAAZZSSXDEH 8.2 Ki 4 Yes
AGFIIERRTNLUMS 8.2 Ki 4 Yes
GQEPEMYIRJCODM 8.2 Ki 2
JQKPNPNQXMEIDL 8.2 Ki 2
PJDNBOOJSSZQPJ 8.2 Ki 2
WHBCDNPPOUFKAB 8.2 Ki 2
IUSJINNBGHLFTG 8.1 Ki 2
RVSCXYLNWULPGJ 8.1 Ki 4 Yes
ZYALYWXELCWDBL 8.1 Ki 4
DTYOTXLNOUBXKR 8.1 Ki 2
QTAUJHKCILRJMG 8.1 Ki 2
ZXMRPSJTSMBYHQ 8.1 Ki 2
UBHYDQAARZKHEZ 8.1 Ki 3
ODHBRFGOHMIIEN 8.1 Ki 2
PBKPCQGTLBWXBQ 8.1 Ki 2
BENDTRBVBYXEFO 8.1 Ki 4
CBSUMJPUYCRHCR 8.1 Ki 2
DJKRSNUQFVHUTB 8.1 Ki 2
FINNTOGAVZWNGL 8.1 Ki 2
FNSGKKGXUCTTRV 8.1 Ki 4
HYPICKIQGZNVCT 8.1 Ki 2
MKMJRTOOXQDCEE 8.1 Ki 2
QQERDUJEEYWVED 8.1 Ki 3 Yes
WZFHAECSSWEURN 8.1 IC50 2
XIRFTMAJUYTWHW 8.1 Ki 2
YHOKBRMLDCDOSC 8.1 Ki 2
ZGFGKYPXTGSMPZ 8.1 Ki 2
MVVKKFHFADVKMW 8.1 Ki 9
FNHGWTOPWMIMCK 8.1 Ki 2
IBDXBPHXQDUOAO 8.1 Ki 2
LAKVEWGOEMZVEF 8.1 Ki 2
LPIYSDRZAIUAIP 8.1 Ki 2
RJXKZVWHSWCCMM 8.1 Ki 2
LOULPFANPPCWQM 8.1 Ki 2
BSDHAHZVUCTDKG 8.1 Ki 2
2D structure