Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
ADHCEOHLWFBYCU 8.5 Ki 2
DWIOHHAGWJCPQF 8.5 Ki 2
ZOTDNNWAQBXDPK 8.5 Ki 2
BOQXUEKBVIXPKQ 8.4 Ki 2
SJTLVMWWYORGEH 8.4 Ki 2
YGGBVTGACIFVRB 8.4 Ki 2
VYEDDDWXKRDQRX 8.4 Ki 4 Yes
HVNNDZMWORMJPO 8.4 Ki 2
ITYMMRKSCDTSQX 8.4 IC50 2
AHOJZWPBIHIALS 8.4 Ki 4 Yes
BENDTRBVBYXEFO 8.4 Ki 4
BXUKKRHEMKVWOY 8.4 Ki 4 Yes
CKIBSEDGQQBNJP 8.4 Ki 2
CQCYZYXYLGEQJN 8.4 Ki 2
CVKJAXCQPFOAIN 8.4 Ki 2
ITYMMRKSCDTSQX 8.4 Ki 2
MEOKXROUBIRKJZ 8.4 Ki 2
OQGUTEKSOMCPOG 8.4 Ki 2
PHSPJQZRQAJPPF 8.4 Ki 2
QYLHCEYSEGRWNL 8.4 Ki 4 Yes
QZAZDEDVSZZTPR 8.4 Ki 4 Yes
ZHNRRDSCSQZYAU 8.4 Ki 2
ZOQAPWIJYCXCQM 8.4 Ki 2
GEYDSVZUDGXVCV 8.4 Ki 3 Yes
HASNZFFRDSPBMJ 8.4 Ki 2
VJSUMPPMFYQOMP 8.4 Ki 2
KZWRVJZTROHTQZ 8.4 Ki 2
YIRWGCANORBOOM 8.4 Ki 3
DCSZPCOOHYVVRY 8.3 Ki 5
YPGRNKJNOSUCLY 8.3 Ki 2
SVBRTHGICYDAAN 8.3 IC50 2
IGFRVSYYVNOZIU 8.3 Ki 2
KADHZYCVSZHNTR 8.3 Ki 2
KSRMXPIAWHFMID 8.3 Ki 4 Yes
SCAVCNGNYHPFKS 8.3 Ki 2
WZRAWTVPOJVPII 8.3 Ki 2
NWZFUZDRGJBHRH 8.3 Ki 2
RTXNVJXREKUAHX 8.3 Ki 2
UKCSSOGUCSSDDR 8.3 Ki 2
WZSXQZNHMKLIIQ 8.3 Ki 2
ZOGKNOVCCQKFNX 8.3 Ki 2
MZCJWLAXZRFUPI 8.3 Ki 2
JCEWQICHOLLRDL 8.3 Ki 4 Yes
OITIJKINXHWSKF 8.3 Ki 4 Yes
YGGBVTGACIFVRB 8.3 Ki 2
GPLGAQQQNWMVMM 8.3 Ki 3
KECSEMPMGDAAQZ 8.3 Ki 4 Yes
PUCXAAZLYORUSG 8.3 Ki 2
DIMAAAZZSSXDEH 8.2 Ki 4
FLLOSWVXSHXQDY 8.2 Ki 2
2D structure