Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
IWBMAAUPHUCYCI 8.5 Kd 20
JASKXIBVQDMBJJ 8.5 Kd 4
KAZRKJFTFFKZLF 8.5 Ki 4 Yes
KCCBFGKNVMTXIQ 8.5 Kd 6
KGGHECZDYBMALC 8.5 Kd 6
KIRWEWNKOWMEBM 8.5 Kd 4
LDXAOQSIBXRCIN 8.5 Kd 6
LKPZDFCAQDGUKZ 8.5 Kd 4
LMBAXHGIFALPQJ 8.5 Kd 4
MODBIBJHAWXYOZ 8.5 Kd 20
MWNWERUECAJGJC 8.5 Kd 6
NNBLASKQLZCYBL 8.5 Kd 4
OBOJTPPADQUWFB 8.5 Ki 4 Yes
OJYUKAHOHYUAHF 8.5 Kd 6
ONVSJLPIADFJKR 8.5 Kd 4
OVYZCEIGUJNWKN 8.5 Kd 4
OZVCVTCZRYMODR 8.5 Ki 4
PCFGLLVVPCPPIG 8.5 Kd 4
PKALTNFRHBJDRH 8.5 Kd 6
QVAKGXNPTKFJST 8.5 Kd 6
RHRPOJKRNUHOJA 8.5 Kd 4
RIDRYHZYVUEBMC 8.5 IC50 2
SLKZDILCMYJAFM 8.5 Ki 2
SRELLSOOXBJTLE 8.5 Kd 4
SYDKBCVMFJSWKD 8.5 Ki 4 Yes
UAFKZBOQJUSIDU 8.5 Kd 4
UHXAVJMDFYIMLP 8.5 Ki 2
USBWQDPYNKDRSV 8.5 Kd 4
UWTPDHDYCBTOMN 8.5 Kd 4
VAICHSCZMSGKPN 8.5 Ki 4 Yes
XNSQSOGNTZGMDA 8.5 Kd 4
XQOLXGFKFIWXQP 8.5 Kd 6
YPAOZTCVMTXDID 8.5 Kd 4
YVJCOHIKEMZVAO 8.5 Kd 4
YVKKYCJACTULJR 8.5 Ki 2
YYXYUTGQFNFTGX 8.5 Kd 4
ZKKBZRDZTBXDKE 8.5 Kd 4
ZYFQYFZOSKEOGJ 8.5 Kd 4
JAPGJDHRYBFKBD 8.5 Ki 2
QJUVWGBVEFRHCN 8.5 Ki 2
BQZCEWUNCDOHHN 8.5 Ki 2
GYJOUMCDNZCUAE 8.5 Ki 2
IKCDGERABUYQOT 8.5 Ki 2
RUMWHMMFUXGDRP 8.5 Ki 2
ZJDRDLAAEMFCJV 8.5 Ki 2
CILDROBPHGWMGB 8.5 Ki 6
NLMXEWVGDSQUMB 8.5 Ki 2
QMAAXHLTCZIRDL 8.5 Ki 4 Yes
RELMLKVZHCPAMI 8.5 Ki 2
RHSFWZWZTDJZPT 8.5 Ki 2
2D structure