Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
NLHDACBKUHRZEW 9.0 Ki 2
WZXBWZLVHBHFDT 9.0 Ki 2
XQRFKDJVDZKQDO 9.0 Ki 3
APQJKSFOISLQFF 8.9 Ki 3
KTSPNBFUARCTGI 8.9 Ki 2
UCAIEVHKDLMIFL 8.9 Ki 4
DTGQAURGKWOQAA 8.9 Ki 2
PESOUNLSPHQJGL 8.9 Ki 2
UCQNMJXTWOYVNH 8.9 Ki 6
OBUQQSWVYWHDKA 8.9 IC50 2
ZQVGMOFPWWNMNB 8.9 Ki 2
GMJQYJUXKUAPMC 8.9 Ki 2
DGRXLTADUFHHBN 8.8 Ki 2
FNMSKRVJSVGVRH 8.8 Ki 2
KTXYACXXINQJMM 8.8 Ki 2
YGGBVTGACIFVRB 8.8 Ki 2
GMTUNRCWXIGLSX 8.8 Ki 2
BCFDOHOQDUCYBU 8.8 Ki 2
IFFHPDKLLFCYAG 8.8 IC50 2
NFCYQBPNSWBYEF 8.8 Ki 4
PEHSVUKQDJULKE 8.8 Ki 2
RRMGPLJQTAJCCP 8.8 Ki 3
SYDQPIHOSLJNHM 8.8 Ki 2
VOXJNIGKOFAGBU 8.8 Ki 2
VZXHLVQQUPAPMN 8.8 Ki 4 Yes
ZSGUUFCXNQUDKV 8.8 Ki 2
JHLZBMJYTQZERX 8.8 Ki 2
ACRVFRPOWNWNAQ 8.8 Ki 2
HBDLBTSITBUDIR 8.8 Ki 2
MJKGHXXXMDVBEW 8.8 Ki 2
OYCZRPQRIZGOTB 8.8 Ki 2
PDKGFOSJNKVHSS 8.8 Ki 2
PXZWAKNYGHYHEV 8.8 Ki 2
QKNQLRSRULGFBA 8.8 Ki 2
QKNQLRSRULGFBA 8.8 Ki 2
WTAQICPSTMPTOD 8.8 Ki 4 Yes
XVGGLWKPTSTHJU 8.8 Ki 2
BJZMQYYHQDWJRH 8.8 IC50 2
CFUHKRLMDNFZED 8.8 Ki 2
ANDYBNKRXGVQGP 8.7 Ki 4
LNKQLDXMYFJALH 8.7 Ki 2
RLDOROHJMZJOFY 8.7 Ki 2
UUTLATQGKXUVDD 8.7 Ki 2
XBIDNEGDXXMQIB 8.7 Ki 2
ZTNPNIPEXVPGCQ 8.7 Ki 2
HZNTWQAMIOKCMC 8.7 IC50 2
VIPAIZRIFZFESY 8.7 Ki 2
WZHAQWFZACLGKI 8.7 Ki 2
XYJMAXNKTLJWRH 8.7 Ki 2
FMTBFJSXJKNLPI 8.7 IC50 2
2D structure