Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
DCQNAFOCXVCDLB 9.2 Ki 2
HKPKDTNLXGOYIC 9.2 Ki 4
LAQGPQNMQRFDIM 9.2 Ki 2
YSFJQETUBNXLQX 9.2 Ki 2
QJFIAPPKZLXTPP 9.2 Ki 2
LQLTVDHLUGEPRE 9.2 Ki 2
BDHLYFHGXMWWJR 9.2 Ki 4 Yes
CRUWXQPBIKVAJO 9.2 Ki 2
LPYJYKOCMFIQCD 9.2 Ki 4 Yes
UWCGILLDYHOPEU 9.2 Ki 2
VUURKLOSWJVNJP 9.2 Ki 2
PPHJOGOEUDGEOR 9.1 Ki 2
BDWXFGZMHKOMCV 9.1 Ki 4 Yes
CAISPEIKDAWTHS 9.1 Ki 7 Yes
CPVIJSYBBQJOPU 9.1 Ki 2
DFVSGZHJSIEEQQ 9.1 Ki 2
IWPSIGJPCATAFI 9.1 Ki 2
JQNSYTMOXNMQTB 9.1 Ki 4
LOMPCAVUANIGGY 9.1 Ki 2
TXFFWCPTQAOPNJ 9.1 Ki 2
YLWKUCPPUFNBEX 9.1 Ki 2
ZRHGDWMRFCDZHY 9.1 Ki 3
KIJIJUXKXSTTLC 9.1 IC50 2
LMCJCKKIGOGRRE 9.1 Ki 2
MDGOMXLQCXHZJE 9.1 IC50 2
NZCBCRNLDOCTQR 9.1 Ki 2
QUZXTJYADOYRDB 9.1 Ki 3
WYKIMPHRITYBHB 9.1 Ki 2
YEXIBZKBLZVZSI 9.1 Ki 2
ASTAPGJBBBKTEX 9.0 Ki 2
OVDJDGHFBGJJHZ 9.0 IC50 2
DCFPUUCKXNHIPZ 9.0 Ki 2
DIKWOUATAGYMJW 9.0 Ki 2
FJWNUBKVWQZAGY 9.0 Ki 4 Yes
HXRQPFYBNJXVTR 9.0 Ki 2
LBAKRWRQQGNMEB 9.0 Ki 2
NQHRYUNHBWFEMY 9.0 Ki 2
ORIYQOUBEPERFH 9.0 Ki 2
PIVRFBAMCBQCDZ 9.0 Ki 3
QSUBPHSKNHPROP 9.0 Ki 2
RGPYWCVMPLKNBH 9.0 Ki 2
UYUUPTYHSLMCNS 9.0 Ki 4 Yes
WCQVQORJCDHBCN 9.0 Ki 2
XTALQXXENKAGEX 9.0 Ki 2
ZKIWXUBGHCOMER 9.0 Ki 2
SIDMDBDAIBEQFI 9.0 Ki 2
DOPOFWDDERLSPU 9.0 Ki 2
CRBTZFVQVOXBBO 9.0 Ki 2
FSAUBGQRVAOUAE 9.0 Ki 2
LUJLISGGFLGFKZ 9.0 Ki 4
2D structure