Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
YLWRKTVVIPNRDE 6.2 Ki 4
DLKAQKCVCFAVIS 6.2 Ki 2
QGWIQIAWOCJRPI 6.2 Ki 6
QUNKNGVNDXGLTG 6.2 Ki 2
YTSCCHQLULFXJD 6.2 Ki 2
QYSFXLSGUKKIAT 6.2 Ki 2
ZFCRJYPCIGHGNV 6.2 Ki 2
JRNUKVFYILMMLX 6.2 Ki 16
MMZLYDNVAYWZLR 6.1 Ki 2
XTWSHHZAQQBXPI 6.1 Ki 2
PREVTMRNRJIUDH 6.1 Ki 2
STDVLBNQKXFBHQ 6.1 Ki 2
BNPPCWFJMXBSSK 6.1 Ki 4
RNUOFCMNVAUGMR 6.1 Ki 2
HWGSTWOVRDYFSO 6.1 Ki 2
MTCUAOILFDZKCO 6.1 IC50 4
QWVFLOZCIRVGKF 6.1 Ki 2
CYECXDNJIMSMBB 6.1 Ki 2
FZFMJBHAXOKONN 6.1 Ki 2
OLHQOJYVQUNWPL 6.1 Ki 2
WYMMYOFAUJTQKL 6.1 Ki 2
AKAAKXSPGNFTCK 6.1 Ki 2
CSQZLIGLFJJGNT 6.1 IC50 2
DZIKZBZBMFPKFM 6.1 Ki 2
WYMMYOFAUJTQKL 6.1 Ki 2
HAOCEOSCGBBHFB 6.1 Ki 4 Yes
MMZLYDNVAYWZLR 6.1 Ki 2
CAIOOXOPQUHZGS 6.0 Ki 2
QXYZJXCNTMMWEO 6.0 Ki 15
DJKJVWJQAVGLHJ 6.0 Ki 8
GXPQVRIHPFBPOG 6.0 Ki 2
UAMIBPKKKLTAKG 6.0 IC50 3
FPUKGJMTLUQGFZ 6.0 Ki 12
BNPPCWFJMXBSSK 6.0 Ki 4
GSYGTVNTZHFQQH 6.0 Ki 2
HMXDWDSNPRNUKI 6.0 Ki 72
KGDAOALFCOEYFT 6.0 Ki 2
KWGDXCJEWFIBAA 6.0 Ki 2
NPSDVAVEQMHDSG 6.0 Ki 2
RFDSGHNJJQPTLS 6.0 Ki 2
2D structure