Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
RETVAMKTDRMQFH 6.5 Ki 2
ZPAHWVAWJGJPSL 6.5 Ki 2
BTBKHELVQIKPDZ 6.5 Ki 2
WDHOIABIERMLGY 6.5 IC50 3
ADEBPBSSDYVVLD 6.5 IC50 6
ADEBPBSSDYVVLD 6.5 IC50 8
FWRAMRVPMYVJMR 6.5 Ki 2
XEMCNPZNSNBIMI 6.5 Ki 4
BKKPIQPFRAPEAY 6.4 IC50 2
HRSYZRFBUGIVHN 6.4 Ki 4
KMFDXNUGIFDFHQ 6.4 Ki 5
PPQJESFHSZPEOS 6.4 Ki 3
RZBPSXCZVILRNE 6.4 Ki 4
HOMWNUXPSJQSSU 6.4 Ki 6
CEQYBPQHHPEWRH 6.4 Ki 4
OARTTZNTSJLCDS 6.4 Ki 4 Yes
CQOZFSIWRBDGOG 6.4 Ki 2
HAIDCJHWMODKNB 6.4 Ki 2
WYRUGBCTQBZIHO 6.4 Ki 5 Yes
YZAHEHXQIMZHAJ 6.4 Ki 5
LMJQZJCJGXDLSR 6.3 Ki 2
QJNCEPWQQYZJCX 6.3 Ki 2
HRIXXYOKKMTERZ 6.3 Ki 2
RXDXCASRBPOFLE 6.3 Ki 2
DTEPKYSLLWLWRZ 6.3 Ki 2
QLLZULWFESFQOY 6.3 Ki 2
ANCFKYJMXNMYNZ 6.3 Ki 3
ICAQZJCLBRKWBG 6.3 Ki 2
IHQGRRRYHOHPFV 6.3 Ki 2
KVHHUZUNLIGTBY 6.3 Ki 10
DHHDEHNHEBYRPQ 6.3 Ki 2
SMVPOIGPHSXRQE 6.3 Ki 4
AZHUBGIQDYLZDQ 6.3 Ki 2
RRWCFKTVVCKJCF 6.3 Ki 2
SSTBBFPDXHDLGH 6.2 Ki 2
XERZUXOKZOACKV 6.2 Ki 4
HAVVGSKWBWZXIO 6.2 Ki 2
HUMDXPQUUMTPFD 6.2 Ki 2
ZWCILIRMPOCMLE 6.2 Ki 2
QTVJIGDYLBRSJM 6.2 Ki 2
DGZLHXBKGBELTQ 6.2 Ki 4
FNEORDYLRZOEEP 6.2 Ki 5
JWDZDXFXHWMSGR 6.2 Ki 3 Yes
KICLSPYVVBSUFF 6.2 Ki 2
PYTFAGDLBOIDSO 6.2 Ki 2
QZUDBNBUXVUHMW 6.2 Ki 39 Yes
REXDQAIKTDDWAC 6.2 Ki 4
SAMYTBZVLLYSKN 6.2 Ki 5
UXQVMDVKHFQOEU 6.2 Ki 5
VFIDGXZRONKQBZ 6.2 Ki 5
2D structure