Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
PLSSBUTVCXDGTH 6.8 Ki 2
ARRCCCIOHBCTKB 6.7 Ki 2
ABYWZGKRJFEJFL 6.7 Ki 2
ISBHYKVAFKTATD 6.7 Ki 2
KBVUBEVDDDEKLM 6.7 Ki 4
ZULPGIJFVSVHRG 6.7 Ki 2
JPDOYLRZYOLBPB 6.7 Ki 3
ZFDZUBGJLKYAKC 6.7 Ki 2
LJHWQMAXBBKMSE 6.7 Ki 2
VWHFISHLSCXQIT 6.7 Ki 4
CJMVJEMHSLDPMO 6.7 Ki 4 Yes
IGZMIXBCHNOMPG 6.7 Ki 2
IMEKNFSOCZJKQI 6.7 Ki 5
YXEZVHWJNRFKSI 6.7 Ki 5
HFJSBLSTDQGNRQ 6.7 Ki 2
QGRLYCYTQSXMLL 6.7 Ki 2
QONNOXSQVWRKPP 6.7 Ki 2
MWULMTACIBZPGN 6.7 Ki 8
LRLYLQHAQNEFGV 6.7 Ki 2
OWUAPKLWWUSEPV 6.7 Ki 2
ILOMBVURTLNCEQ 6.7 Ki 2
DMZILZFFWINIES 6.6 Ki 4
MSGVDWYIUWBRPF 6.6 Ki 4
NDDYCWJCTGXGIS 6.6 Ki 2
KWWHIDCVULQSFZ 6.6 Ki 2
RETVAMKTDRMQFH 6.6 Ki 2
SXNOWQCFHNZUIX 6.6 Ki 4
UJMUXUJLIHKBEA 6.6 Ki 4 Yes
YMFHXRKTKHBRIX 6.6 Ki 4 Yes
UYMBIBLZLAJMQD 6.6 Ki 2
XJPIMYAKYUJUQV 6.6 Ki 4
YTCGNPGLMAECND 6.6 Ki 2
DTDLOHYXZTWBHO 6.6 Ki 2
FFUYAMBLAURQHK 6.6 Ki 4
QFOKEUVZRMQKAH 6.6 Ki 2
QQICDAPFTVTGQB 6.6 Ki 4
UHHNLJHQYLBBSB 6.6 Ki 4
WURDXGJSSCNLKT 6.6 Ki 2
WKMOBAVFRIULDB 6.5 IC50 2
SGHHKDMDVKJWOL 6.5 Ki 2
ZRTFTZCKJUNZIU 6.5 IC50 4
ZTOUOCYMUXLHOP 6.5 Ki 2
DPJNKUOXBZSZAI 6.5 Ki 4
XYXNDRMGQIINHD 6.5 Ki 3
GSRZQXGOVFSDAD 6.5 Ki 4
HPYFHGSUPFFSGC 6.5 Ki 2
OUEZWZJJIKBFFV 6.5 Ki 5
URSKGEZFWCRYMD 6.5 Ki 3 Yes
YQXATUVEKBYLGN 6.5 Ki 3
KTBGOCBJUUOAMQ 6.5 Ki 2
2D structure