Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
OZVCVTCZRYMODR 7.0 Ki 4
UXYHRAYDBQKHHN 7.0 Ki 2
XOGYORIOPYTSDW 7.0 Ki 4
ICIGFIHEQAKGAX 7.0 Ki 2
IMIDSGXDTGNBGW 7.0 Ki 2
SNEWMZUDBQVWAO 7.0 Ki 2
CSDCGOJSTHVMSW 7.0 Ki 2
JREXJAZIYYZNSO 7.0 Ki 3
NMHISCWMQDLSTP 7.0 Ki 2
KTIHAAVUVHUODX 7.0 Ki 2
MMXFVUGZZAXQNG 7.0 Ki 2
UREJDUPKGMFJRU 7.0 Ki 17
JXLGDCHDFPYUFA 7.0 Ki 2
NCFNOILQWULHEZ 7.0 Ki 2
HLLYNFMNKJGCNN 7.0 Ki 4
VQTUECJHHAWNKZ 7.0 Ki 2
SBAPLMPNRPQJSQ 6.9 Ki 2
CSHFHSIPMYFXHR 6.9 Ki 2
PPQJESFHSZPEOS 6.9 Ki 2
CRGOWMIZBWIMTB 6.9 Ki 2
FRUMSZUUBXPHHF 6.9 Ki 4 Yes
HBSZYLFXYCHZJR 6.9 Ki 4
SAKVKDBLCRHLAV 6.9 Ki 4 Yes
WNDPQJQMFPORJY 6.9 Ki 2
HVBQQFJIXGEUPB 6.8 Ki 2
NLVYWCRLGFDESU 6.8 Ki 2
OQBDNCOEWGLQTE 6.8 Ki 2
ULVWQSSQQHJQPK 6.8 Ki 2
LTHPEUUEWQVVRQ 6.8 Ki 2
QLLZULWFESFQOY 6.8 Ki 2
VZBVZINFDHFRML 6.8 Ki 2
BFLDMZUQHIXFAK 6.8 Ki 4
HGCSDFHPKCOZNX 6.8 Ki 2
LJDQVOLRQLNUCX 6.8 Ki 4
MBUVEWMHONZEQD 6.8 Ki 17 Yes
AQIRLJIMBMOXCB 6.8 Ki 2
HTLDHQKBLGJBRF 6.8 Ki 2
IHWMDXVSMHTLOY 6.8 Ki 4
RIDMUSSNFOKJBO 6.8 Ki 4
QJEBESRHAPCDHQ 6.8 Ki 2
MJRWQKDJTQKTMJ 6.8 Ki 3
UKIGXRPAJQOYHR 6.8 Ki 2
HREUGOAZLRNTEM 6.8 Ki 2
MVTKOPGIBNCWRJ 6.8 Ki 4
PMQRGOWDOYXFIQ 6.8 Ki 4
WQWHPPMEWVYOCN 6.8 Ki 4
DFFKMCAWTADECS 6.8 IC50 2
KNIPHGXUVWAHCN 6.8 Ki 3
UGXJCFJERJLZKI 6.8 Ki 2
HGLGWLWXYRAXPK 6.8 Ki 3
2D structure