Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
RBJDHCDYYMNJHT 7.3 Ki 2
XKAQYEAHVGQUFQ 7.3 Ki 2
ZUIOKZVLMBWAPI 7.3 Ki 2
IHDFTEVCMVTMSP 7.3 Ki 2
UZFUMFWJEGINFP 7.3 Ki 2
QKDDJDBFONZGBW 7.3 Ki 5
FDGXVDUYFWJNRM 7.3 Ki 6
HZJHXNKBUJZZBB 7.3 Ki 2
NLDYNKODZYDSNC 7.3 Ki 4 Yes
ZLULVVLDDHMAFR 7.3 Ki 2
ZMYWSFVTVVHGEG 7.3 Ki 2
JPDOYLRZYOLBPB 7.2 Ki 3
PARJGQCKHQBNLB 7.2 Ki 2
PCLYKAGGELJIIV 7.2 Ki 4
ACQBHJXEAYTHCY 7.2 Ki 5
FNLKLDDVROBECF 7.2 Ki 2
KMJZIGCXRSSFHL 7.2 Ki 2
PRWLDKKWXOINJS 7.2 Ki 2
RWWMQYYGHIHOGU 7.2 Ki 2
XNQIOISZPFVUFG 7.2 Ki 2
XOTVIUDNDAPPIB 7.2 Ki 2
NYERXTAQHGNTEO 7.2 Ki 2
RHFLZSUIVOSCKT 7.2 Ki 6
YVGCLDBDDBQLIK 7.2 Ki 2
KPAJJCMZSUJZLQ 7.2 Ki 2
MURRAGMMNAYLNA 7.2 Ki 2
OXKMEPWPNZHEEF 7.2 Ki 2
WUWSDBLNZJIRHW 7.2 Ki 2
AUMQJULFKZREJZ 7.2 Ki 2
DFXVOYQWLICYQI 7.2 Ki 2
IQMRECYOUIKYGG 7.1 Ki 2
KUWPQNYVWRUDNF 7.1 Ki 2
UVYNECUSQBZMSD 7.1 Ki 2
WJEAZFGKRWLAIJ 7.1 Ki 2
CUMDGRCUGGUZMS 7.1 Ki 2
GRWARSULWXLZOY 7.1 Ki 2
HNLNXYUSMGCHFW 7.1 Ki 4 Yes
MBVVVQZOMZFVJF 7.1 Ki 4 Yes
PSFPFXQRWTYKOH 7.1 Ki 2
UOBXGIKOILQPJJ 7.1 Ki 2
VTMJTHCQLMVWGT 7.1 Ki 4
CPWCCIJQANDZQE 7.1 Ki 2
ADCBAOTWERXLAP 7.1 Ki 6
HXRBAVXGYZUSED 7.1 Ki 2
LMPVKITTWDPCLI 7.1 Ki 2
HBOJWAYLSJLULG 7.1 Ki 5
XTZKOGDXCXHQKA 7.0 Ki 2
UKHIUWLEJYNXSB 7.0 Ki 2
BNXNWRSVYQHTOH 7.0 Ki 12
MKSDMOQTAOJLSE 7.0 Ki 4 Yes
2D structure