Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
ZXIIHOHNYIUMNQ 7.6 IC50 2
UYXWQSZIUMRFIW 7.6 Ki 2
KIDYDIXDUYDRBZ 7.6 Ki 2
SZALSWFXFHISRB 7.6 Ki 2
ZZPQCQWVWDUPSI 7.6 Ki 2
BOAJEIFQZOFOCK 7.5 Ki 2
BRKDRAMGEIRGGU 7.5 Ki 2
DXJUCAUQIHNOAF 7.5 Ki 6
PCLYKAGGELJIIV 7.5 Ki 4
UESRDXOTUAFPQL 7.5 Ki 2
BJWZNXSSJMLUNB 7.5 Ki 4 Yes
SWTVGVLYEISYND 7.5 Ki 5
UWWLHNUJLKTVOD 7.5 Ki 2
LZUBTFVEEDSMJZ 7.5 Ki 2
MJTKHTWGWXGNME 7.5 Ki 2
WPDUKOOPOVGUGG 7.5 Ki 2
WWTASRSHEGBDMT 7.5 Ki 2
SHQNNJIERWMYHK 7.5 Ki 2
ZTRXSQAFMVDLBU 7.5 Ki 2
USFDQTKOPQREEH 7.5 Ki 2
HJLCHLAAXMALNR 7.5 Ki 2
LMFNLINKCDGRTE 7.5 Ki 2
NESASFDNMLPZIR 7.5 Ki 2
SGHHKDMDVKJWOL 7.5 Ki 2
JGRNPFVRYKMKOL 7.4 Ki 2
KXTUUFGXZCWFKF 7.4 Ki 2
LVKNXJNGRXMDCY 7.4 Ki 4
HIZHUDHSNMVOFW 7.4 Ki 2
LCRAAWGCGKXFMG 7.4 Ki 2
CWKGVKHDADMKBI 7.4 Ki 2
NOSCCMUAADBXHH 7.4 Ki 2
AFJWXHZYSMRBOR 7.4 Ki 2
AVZAABIFUPTQRO 7.4 Ki 2
CGIBXEHRRLWSKY 7.4 Ki 2
FJWJHKWEIJMGPV 7.4 Ki 2
MFUXHAFVFJVNEU 7.4 Ki 2
STQJDUUWFXFIQR 7.4 Ki 2
BYUXJHZOSYXPSS 7.4 IC50 2
HGXALICWKOVEQW 7.4 Ki 2
HUDWMNWXZIMODJ 7.4 IC50 2
JDUPATOWYGPGEY 7.4 Ki 2
YTYOOWFUEIQRHQ 7.4 Ki 2
AYKJGACMCQMMAW 7.4 Ki 2
INWLSQYDDFJBQN 7.4 Ki 2
XOWPFAUTGJEGMK 7.4 Ki 2
BOQXUEKBVIXPKQ 7.4 Ki 2
RNAMYOYQYRYFQY 7.3 Ki 3
FYQWSOGFMUPHGU 7.3 Ki 2
JGXWDNPDGKMFIY 7.3 Ki 2
SAEILUJHGHNPAN 7.3 Kd 4
2D structure