Target Details
UniProt ACQ9Y5N1
Gene SymbolHRH3
Protein NameHistamine H3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 740
  • Clinical molecules 71
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (740)
InChIKey pChEMBL Type Targets Clinical
OXJGPZFAZUEPIX 10.4 Ki 6
BCSPALWWQLYRIR 10.0 Ki 2
CNMDDAFIBJNBFQ 9.8 Ki 2
DQUUMUHVZGIZNI 9.8 Ki 2
YOQCIOKHHDUPPQ 9.8 IC50 2
DZMTUSAQZVLLBN 9.7 Ki 2
SPKOQCHHYOCMGR 9.7 Ki 2
DFTFGLPAHCOAEP 9.7 Ki 3
IFLIPLANALCYLX 9.6 Ki 2
IVVRZZSSLSFZID 9.6 Ki 2
REXVRCXDIWIKGL 9.6 Ki 4 Yes
YANGEESWIGIKOP 9.6 Ki 4 Yes
YANGEESWIGIKOP 9.6 Ki 7 Yes
MYSZKGRXICYNIZ 9.6 Ki 2
VGSYEFOBFMUWGO 9.6 Ki 6
OYWQMDWRCCYZOE 9.6 Ki 4
UBKCIYMLUUFSDB 9.5 Ki 2
NCHOEXFBJYYHOD 9.5 Ki 2
AWKFJGDSZGEFRY 9.5 Ki 4 Yes
FZTMDWIJTHPEMP 9.5 Ki 4
GLSCKISDOLHCSX 9.5 Ki 2
GLSCKISDOLHCSX 9.5 Ki 2
MHAQFNSWCQLYOT 9.5 Ki 2
IBPWGZKZWJYGLA 9.5 Ki 3
ILIWVAFIMXCJTB 9.5 Ki 2
AQQFXOLTZFTABW 9.4 Ki 6
JHZTZJQZFCCJBJ 9.4 Ki 2
RDPSEAZFXPEZMP 9.4 IC50 2
GPZMWOXSIRVXQW 9.4 Ki 8
GQWSXILTLUTBAJ 9.4 Ki 4 Yes
IMKMPTLRTHMERW 9.4 Ki 4 Yes
OWYPWYDPIBLTEG 9.4 Ki 2
UUYDLXMNWLLYQV 9.4 Ki 4 Yes
XHHDACAEDLRJOJ 9.4 Ki 5
YZSDHSPCNCYZKJ 9.4 IC50 2
PQPVHIHIJVIEQG 9.4 Ki 6
KFHYZKCRXNRKRC 9.3 Ki 2
MCNGUYXRBCIGOV 9.3 Ki 2
QYDDQJVHZBTEMT 9.3 Ki 2
CVFUNUQUAWLUGT 9.3 Ki 2
DRLFMBDRBRZALE 9.3 Ki 4
QYAXGGUCDQSHIT 9.3 Ki 4 Yes
RHTRBRRAADVASO 9.3 Ki 4
VGLVSBTUAYHUEF 9.3 Ki 2
YSFJQETUBNXLQX 9.3 Ki 2
CXRCFQKCULIFAC 9.3 Ki 2
CIAWHNGOFJZBCL 9.2 Ki 5
GMAJNYRLILNPJN 9.2 Ki 3
WBLFYMQYQYGVGK 9.2 Ki 2
AGSWPZXGFSITHZ 9.2 Ki 2
2D structure