Target Details
| UniProt AC | Q9Y5K2 |
|---|---|
| Gene Symbol | KLK4 |
| Protein Name | Kallikrein-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 8.18
Associated Diseases (1)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WONGRAWCJSVHOJ
|
10.0 | Ki | 5 | — | |
KHTRPJFHQNRISN
|
9.4 | Ki | 5 | — | |
WBFBQDAAAKLBHB
|
8.8 | Ki | 2 | — | |
RMJHMNZGTJDKCS
|
8.5 | IC50 | 4 | — | |
VRMZLUPLYRHORK
|
8.1 | Ki | 6 | — | |
CTDHLROQTKJDLK
|
7.9 | IC50 | 4 | — | |
MWBNFSUYTZMPST
|
7.8 | IC50 | 3 | — | |
AOMZQHHLSHFCGW
|
7.7 | Ki | 2 | — | |
IVGMDANEFALECQ
|
7.4 | IC50 | 5 | — | |
WYCVSPRVSFUVMA
|
7.4 | IC50 | 3 | — | |
CSTAEACZUNFQMP
|
7.1 | IC50 | 3 | — |