Target Details
| UniProt AC | Q9Y572 |
|---|---|
| Gene Symbol | RIPK3 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF12721 (RHIM) |
Summary
- Multi-target molecules 67
- Clinical molecules 2
- Avg pChEMBL 7.02
KEGG Pathways (5)
Active Molecules (67)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FNHKPVJBJVTLMP
|
6.4 | Kd | 29 | — | |
MEWQFVCNRWMTNX
|
6.4 | IC50 | 2 | — | |
LPFWVDIFUFFKJU
|
6.4 | Kd | 9 | — | |
XTCHKTGNNBBKHW
|
6.4 | IC50 | 2 | — | |
CKZNIIZTVZQXIP
|
6.4 | IC50 | 2 | — | |
XFXAMCQJMNCCHZ
|
6.4 | IC50 | 2 | — | |
YKOORZPNFGWYGV
|
6.3 | IC50 | 2 | — | |
ZGBAJMQHJDFTQJ
|
6.3 | Kd | 15 | — | |
JWDPCUJHMUSEKL
|
6.3 | IC50 | 2 | — | |
CVWXJKQAOSCOAB
|
6.2 | IC50 | 35 | — | |
LNMRSSIMGCDUTP
|
6.2 | Kd | 13 | — | |
SNRUTMWCDZHKKM
|
6.2 | Kd | 4 | — | |
UEHMGSTWWBKBBG
|
6.1 | Kd | 2 | — | |
CMJCXYNUCSMDBY
|
6.0 | Kd | 15 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |