Target Details
| UniProt AC | Q9Y572 |
|---|---|
| Gene Symbol | RIPK3 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF12721 (RHIM) |
Summary
- Multi-target molecules 67
- Clinical molecules 2
- Avg pChEMBL 7.02
KEGG Pathways (5)
Active Molecules (67)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OJUQYRUOIGTYSD
|
9.5 | IC50 | 2 | — | |
UGTLDBJIOSYXRR
|
9.5 | IC50 | 2 | — | |
PHXJVRSECIGDHY
|
8.8 | IC50 | 59 | — | |
ZCDBTQNFAPKACC
|
8.7 | IC50 | 3 | — | |
UFWJGUUHERHCOL
|
8.5 | IC50 | 3 | — | |
AQSSMEORRLJZLU
|
8.5 | Kd | 34 | Yes | |
BGDMMVIAARSUKG
|
8.1 | Kd | 2 | — | |
BPKSNNJTKPIZKR
|
8.1 | IC50 | 2 | — | |
QMILKASSWHCTOF
|
8.1 | IC50 | 4 | — | |
IVRXNBXKWIJUQB
|
8.0 | Kd | 10 | — | |
BXJAJCQUQYZMSO
|
7.8 | IC50 | 2 | — | |
XLOGLWKOHPIJLV
|
7.8 | IC50 | 3 | — | |
WVXNSAVVKYZVOE
|
7.7 | IC50 | 92 | — | |
SZNYUUZOQHNEKB
|
7.7 | IC50 | 7 | — | |
VMXQAQDFSBPASA
|
7.5 | Kd | 2 | — | |
DGOLQKDWHOHSFK
|
7.4 | Kd | 2 | — | |
WFWVJTWOJNJWJW
|
7.3 | Kd | 2 | — | |
DSKYHEJWWIBREA
|
7.1 | Kd | 8 | — | |
GDANGPXOFKSTJT
|
7.1 | IC50 | 2 | — | |
AVPUTQITOHDIOV
|
7.1 | Kd | 2 | — | |
SDSQERWTMKMZLA
|
7.1 | Kd | 2 | — | |
XYFPWWZEPKGCCK
|
7.1 | Kd | 34 | — | |
KVVWSWZRLJGEJZ
|
7.1 | IC50 | 2 | — | |
UWXSAYUXVSFDBQ
|
7.1 | Kd | 6 | — | |
ZQSZVECJMJELSV
|
7.0 | IC50 | 2 | — | |
RHGWZRPWVUJSPD
|
7.0 | Kd | 2 | — | |
OJFKUJDRGJSAQB
|
7.0 | Kd | 17 | — | |
LEKAQKZSVPRISA
|
7.0 | Kd | 2 | — | |
OUMWMQOMQTXCGS
|
6.9 | IC50 | 2 | — | |
DWKAWEVEZABLJA
|
6.9 | Kd | 2 | — | |
LZTBBNONIGEIKH
|
6.9 | Kd | 2 | — | |
PZBUOCXBGCVSAF
|
6.9 | Kd | 2 | — | |
NENVTQZTFIQRHK
|
6.9 | IC50 | 2 | — | |
BVFILFYBSTWUCR
|
6.9 | Kd | 2 | — | |
UMLPCOVOJFEKRE
|
6.8 | IC50 | 2 | — | |
WANGYKOAXRTHJB
|
6.8 | Kd | 2 | — | |
CXQHYVUVSFXTMY
|
6.8 | Kd | 154 | — | |
UQRCJCNVNUFYDX
|
6.8 | Kd | 27 | — | |
OBSFXHDOLBYWRJ
|
6.7 | IC50 | 7 | Yes | |
BXVRODNTVCIXSZ
|
6.7 | Kd | 2 | — | |
DKNUPRMJNUQNHR
|
6.6 | Kd | 33 | — | |
BFSMGDJOXZAERB
|
6.6 | IC50 | 33 | — | |
WANGYKOAXRTHJB
|
6.6 | Kd | 2 | — | |
WKHMETWKHWYTEE
|
6.6 | IC50 | 2 | — | |
NFUVBUNETZNUIB
|
6.5 | Kd | 2 | — | |
KUDLEBZUOBVRGB
|
6.5 | IC50 | 2 | — | |
WOSKHXYHFSIKNG
|
6.5 | Kd | 24 | — | |
DKZYXHCYPUVGAF
|
6.5 | Kd | 112 | — | |
HVXKQKFEHMGHSL
|
6.4 | Kd | 21 | — | |
JTQDNMQENCMSFD
|
6.4 | IC50 | 2 | — |