Target Details
| UniProt AC | Q9Y4K4 |
|---|---|
| Gene Symbol | MAP4K5 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 280
- Clinical molecules 35
- Avg pChEMBL 6.9
Active Molecules (280)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJLAWZDWDVHWOW
|
6.1 | Kd | 4 | — | |
VCSQVKQFGYRGEH
|
6.1 | Ki | 13 | — | |
VXYDJXMHISGSDA
|
6.1 | Ki | 59 | — | |
WVFWTUJEHMVUBG
|
6.1 | Ki | 25 | — | |
XYXLUJQBBIBJFV
|
6.1 | Ki | 36 | — | |
YACXOXQTGJXYNX
|
6.1 | Ki | 11 | — | |
ZLVOTRRGLSDLPF
|
6.1 | Ki | 36 | — | |
PBCZSGKMGDDXIJ
|
6.1 | Kd | 68 | Yes | |
YABJJWZLRMPFSI
|
6.1 | Kd | 34 | — | |
RYYNGWLOYLRZLK
|
6.0 | Kd | 45 | — | |
HVXKQKFEHMGHSL
|
6.0 | Kd | 21 | — | |
MPVGZUGXCQEXTM
|
6.0 | Kd | 61 | Yes | |
HHCBMISMPSAZBF
|
6.0 | IC50 | 23 | — | |
AGYRJOAGMDIFKL
|
6.0 | Ki | 17 | — | |
AOBLBPWPSKBHSI
|
6.0 | Ki | 55 | — | |
AQQWWOMMPDCTLW
|
6.0 | Ki | 10 | — | |
BIIVYFLTOXDAOV
|
6.0 | Ki | 31 | — | |
FXXMEMJTLOATRB
|
6.0 | Ki | 5 | — | |
HTROFVQKJODSCL
|
6.0 | Ki | 11 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KWSZYBNXNYRQCC
|
6.0 | Ki | 21 | — | |
MADCXGNPDBWPLM
|
6.0 | Ki | 25 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
OETCTXGISYWYMV
|
6.0 | Ki | 7 | — | |
WKEYMNLZBZKLOG
|
6.0 | Ki | 14 | — | |
XBAIEEJJCJHBDL
|
6.0 | Ki | 17 | — | |
XGMWRIIMIJPGBH
|
6.0 | Ki | 10 | — | |
XSRHBCYNCKAFKS
|
6.0 | Ki | 45 | — | |
XXSPHNFKLDJDAK
|
6.0 | Ki | 26 | — |