Target Details
| UniProt AC | Q9Y4K4 |
|---|---|
| Gene Symbol | MAP4K5 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 280
- Clinical molecules 35
- Avg pChEMBL 6.9
Active Molecules (280)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XNEPVLVYFUGJLF
|
6.7 | Ki | 27 | — | |
QKNBRNSGPNCARD
|
6.7 | IC50 | 9 | — | |
VAARYSWULJUGST
|
6.6 | Kd | 119 | Yes | |
RVSSNRBUPQUIEG
|
6.6 | IC50 | 5 | — | |
CFIBXVQLBVNOHW
|
6.6 | Ki | 64 | — | |
DFMCXVONDDGQIY
|
6.6 | Ki | 66 | — | |
DJLORVJVWIBDME
|
6.6 | Ki | 24 | — | |
DQPYZHUAILXFJI
|
6.6 | Ki | 27 | — | |
GWMATETWMAQOFL
|
6.6 | Ki | 36 | — | |
GXKYSFQMTTZPGW
|
6.6 | Ki | 7 | — | |
HXHAJRMTJXHJJZ
|
6.6 | Ki | 52 | Yes | |
NJPWCTYVEJIQBM
|
6.6 | Ki | 72 | — | |
RITAVMQDGBJQJZ
|
6.6 | Ki | 33 | — | |
SRONQUHCRFZABC
|
6.6 | Ki | 28 | — | |
TUJUZVJICDSNLY
|
6.6 | Ki | 19 | — | |
UVZVWLFSZNPMBS
|
6.6 | Ki | 17 | — | |
XPHWIERLJBFPFV
|
6.6 | Ki | 69 | — | |
YUOWJICKAJQZLS
|
6.6 | Ki | 35 | — | |
ZQUSFAUAYSEREK
|
6.6 | Ki | 7 | — | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
CKVWQORGCCEYHS
|
6.5 | Ki | 50 | — | |
GHPFSYCYZJKVDZ
|
6.5 | Ki | 18 | Yes | |
MLDQJTXFUGDVEO
|
6.5 | Ki | 85 | Yes | |
MVJMMLFMPWITEJ
|
6.5 | Ki | 110 | — | |
NLUPJKQOKWBWFC
|
6.5 | Ki | 69 | — | |
PKCDDUHJAFVJJB
|
6.5 | Ki | 13 | — | |
PLHUMPJXRHMFFR
|
6.5 | Ki | 28 | — | |
QXKKPVVOOWBLND
|
6.5 | Ki | 8 | — | |
UAQJVFADAYIBGC
|
6.5 | Ki | 23 | — | |
ODPGGGTTYSGTGO
|
6.5 | Kd | 153 | — | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
OSVUGUHRKMMBSE
|
6.4 | Kd | 170 | — | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
IOBVCHJTLVPPBR
|
6.4 | Ki | 39 | — | |
JAMDNXUAYUHJLJ
|
6.4 | Ki | 40 | — | |
JPCWMTOYDYYXLS
|
6.4 | Ki | 7 | — | |
JTRNNNVASYCTLO
|
6.4 | Ki | 14 | — | |
KIUHBHFVVQQALF
|
6.4 | Ki | 9 | — | |
KJVWCDAPVMWKLJ
|
6.4 | Ki | 20 | — | |
KTWBYGUSEYSRND
|
6.4 | Ki | 28 | — | |
LCHCSKHPVCDXAU
|
6.4 | Ki | 30 | — | |
OWDRQHVEJIYVOI
|
6.4 | Ki | 47 | — | |
PSCJSWRVCKUMSL
|
6.4 | Ki | 35 | — | |
QTQUAHGXBLFSCH
|
6.4 | Ki | 10 | — | |
SBFPHSVZEXSHTL
|
6.4 | Ki | 62 | — | |
UTMRCMCLMBDPNW
|
6.4 | Ki | 10 | — | |
VUHZDNOPEVGHEO
|
6.4 | Ki | 29 | — | |
XAHJIRNRDAKTEF
|
6.4 | Ki | 18 | — | |
CVWXJKQAOSCOAB
|
6.4 | Kd | 35 | — |