Target Details
| UniProt AC | Q9Y4K4 |
|---|---|
| Gene Symbol | MAP4K5 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 280
- Clinical molecules 35
- Avg pChEMBL 6.9
Active Molecules (280)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GMYYMEOGFRKSFS
|
7.0 | Ki | 29 | — | |
IJRBJCMLWLFMIN
|
7.0 | Ki | 17 | — | |
ILUGAYBMBIJXHC
|
7.0 | Ki | 9 | — | |
KEZAHTDTAWUZDU
|
7.0 | Ki | 8 | — | |
NZVDDFRUBIEKLV
|
7.0 | Ki | 20 | — | |
OUJZYQBEFNDJQN
|
7.0 | Ki | 71 | — | |
SMRWVXLSRJWVBF
|
7.0 | Ki | 25 | — | |
TVUWQDLBEOZVOU
|
7.0 | Ki | 41 | — | |
WVXNSAVVKYZVOE
|
7.0 | IC50 | 92 | — | |
XMGFTZYNTYNOOJ
|
7.0 | Ki | 10 | — | |
XXJWYDDUDKYVKI
|
7.0 | Kd | 52 | — | |
YMIJUBCSOKSFRU
|
7.0 | Ki | 87 | — | |
GEGCXGMFUYJULA
|
6.9 | Ki | 30 | Yes | |
HOYRWTWZUFFACV
|
6.9 | Ki | 28 | — | |
IAKGNUWZPSPEKU
|
6.9 | Ki | 19 | — | |
JSDGKSMNPHJDFK
|
6.9 | Ki | 35 | — | |
LCGSWTFWYNYUKS
|
6.9 | Ki | 26 | — | |
MZDKLVOWGIOKTN
|
6.9 | Ki | 80 | — | |
RJZDECGDCKOHBV
|
6.9 | Ki | 70 | — | |
RWKDVIAVTRRJIR
|
6.9 | Ki | 23 | — | |
XAYDUCQADQTDGX
|
6.9 | Ki | 12 | — | |
ZXLFIHLBHMLHFJ
|
6.9 | Ki | 31 | — | |
AAYZTFLAQXDFOL
|
6.8 | Ki | 11 | — | |
ACSYKUPGCXYRRO
|
6.8 | Ki | 26 | — | |
AUDNGNGLLRZLDR
|
6.8 | Ki | 33 | — | |
CHTMRWQLNNRRFJ
|
6.8 | Ki | 70 | — | |
CNQGNADBGYCKKV
|
6.8 | Ki | 25 | — | |
GDYZFFBMSBDTAA
|
6.8 | Ki | 60 | — | |
HRZOUBQYVUXBNS
|
6.8 | Ki | 38 | — | |
LRZYYIZFBXFSJB
|
6.8 | Ki | 69 | — | |
OAVGBZOFDPFGPJ
|
6.8 | Ki | 42 | Yes | |
OWRXHGAFWZFFCW
|
6.8 | Ki | 113 | — | |
QNUKRWAIZMBVCU
|
6.8 | Ki | 46 | — | |
QYZOGCMHVIGURT
|
6.8 | Kd | 26 | Yes | |
XNWKXXIGSPPPBH
|
6.8 | Ki | 31 | — | |
XUFLBSMTYMFOQH
|
6.8 | Ki | 43 | — | |
YEHCNYAQEBQCCS
|
6.8 | Ki | 74 | — | |
YEPNVBNYCRGZRX
|
6.8 | Ki | 26 | — | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
IAYGCINLNONXHY
|
6.7 | Kd | 50 | — | |
KOZFSFOOLUUIGY
|
6.7 | Kd | 88 | Yes | |
HEUSUIRCBWROMH
|
6.7 | Ki | 64 | — | |
JSKUWFIZUALZLX
|
6.7 | Ki | 33 | — | |
LACOMQAWPSFXQC
|
6.7 | Ki | 27 | — | |
LRLDYTTWQIFWBD
|
6.7 | Ki | 25 | — | |
NERQMDXDVAZVNX
|
6.7 | Ki | 13 | — | |
NXNQLECPAXXYTR
|
6.7 | Ki | 29 | — | |
QPORZABOFXPRHM
|
6.7 | Ki | 18 | — | |
RFBPWKMQWSIPEO
|
6.7 | Ki | 28 | — | |
VIJBEUTVNBPGIU
|
6.7 | Ki | 19 | — |