Target Details
| UniProt AC | Q9Y4K4 |
|---|---|
| Gene Symbol | MAP4K5 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 280
- Clinical molecules 35
- Avg pChEMBL 6.9
Active Molecules (280)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IBPSHHSPUPWXHN
|
7.5 | Ki | 6 | — | |
LPILBMJJRGTKOQ
|
7.5 | Ki | 27 | — | |
OGNYUTNQZVRGMN
|
7.5 | Ki | 16 | Yes | |
PUPCRRRSBUYJAD
|
7.5 | Ki | 44 | Yes | |
QONPPIZSNSSCSK
|
7.5 | Ki | 45 | Yes | |
UDFDIIVNIYWXDM
|
7.5 | Ki | 74 | — | |
ZGGIYFOLDBTZIL
|
7.5 | Ki | 27 | — | |
APPXQUDJLJXULP
|
7.4 | IC50 | 47 | — | |
GXJSLIOOPZRPEV
|
7.4 | Ki | 34 | — | |
RWEHAHIEUDLKGT
|
7.4 | Ki | 33 | — | |
SLKCVFPEQGHNSI
|
7.4 | Ki | 29 | — | |
WINHZLLDWRZWRT
|
7.4 | Kd | 201 | Yes | |
UIARLYUEJFELEN
|
7.4 | Kd | 289 | Yes | |
CXQHYVUVSFXTMY
|
7.3 | Kd | 154 | — | |
KTEIFNKAUNYNJU
|
7.3 | Ki | 48 | — | |
ZBNZXTGUTAYRHI
|
7.3 | Kd | 102 | Yes | |
AZTMYWWWILJAKW
|
7.3 | Ki | 16 | Yes | |
CXBBWVXSZINRCS
|
7.3 | Ki | 41 | — | |
LSLPDHNUWRDOGC
|
7.3 | Ki | 25 | — | |
OADRBDVURCEKRP
|
7.3 | Ki | 44 | — | |
RIUZPIBUSOHUKF
|
7.3 | Ki | 23 | — | |
SEVCBWKJSOLMNQ
|
7.3 | Ki | 38 | — | |
UQJQNZHGEVLHST
|
7.3 | Ki | 15 | — | |
UWDBNTXEKYRMSG
|
7.3 | Ki | 26 | — | |
WDARYLSSWBWVCU
|
7.3 | Ki | 49 | — | |
ZWVZORIKUNOTCS
|
7.3 | Ki | 69 | — | |
BHSOPYVVEZFHDB
|
7.2 | Ki | 25 | Yes | |
BSFNGHCTZDCQBF
|
7.2 | Ki | 93 | — | |
DLWMVUDMPMKGEE
|
7.2 | Ki | 24 | — | |
FDVSOQRNTAPCHB
|
7.2 | Ki | 40 | — | |
PUYIXDDMOUMMRR
|
7.2 | Ki | 27 | — | |
YDWMUCKJUNLURC
|
7.2 | Ki | 24 | — | |
YWTBGJGMTBHQTM
|
7.2 | Ki | 65 | — | |
DKZYXHCYPUVGAF
|
7.2 | Kd | 112 | — | |
BGYVWFZMYBWCNY
|
7.1 | Ki | 30 | — | |
DZSUJUOJJJCWGG
|
7.1 | Ki | 55 | Yes | |
FUMCKNCUEAQHCV
|
7.1 | Ki | 103 | — | |
GCBJDOWIQHMCMR
|
7.1 | Ki | 84 | — | |
GHMRUNOHAHJNNA
|
7.1 | Ki | 29 | — | |
KTEIFNKAUNYNJU
|
7.1 | Kd | 114 | — | |
OLUKILHGKRVDCT
|
7.1 | Ki | 44 | Yes | |
OYONTEXKYJZFHA
|
7.1 | Kd | 69 | Yes | |
PNKALLUVKOKYHZ
|
7.1 | Ki | 32 | — | |
QKPLUKMJEKRAJD
|
7.1 | Ki | 30 | Yes | |
UMTWTCVTRDYHQQ
|
7.1 | Ki | 56 | — | |
GCIKSSRWRFVXBI
|
7.1 | Kd | 109 | Yes | |
NXSJMRCTGYTSTK
|
7.1 | Kd | 200 | — | |
DORZPJWJOBMQKC
|
7.0 | IC50 | 9 | — | |
BLQYVHBZHAISJM
|
7.0 | Ki | 54 | — | |
FLEAYYMORDPWAJ
|
7.0 | Ki | 90 | — |