Target Details
| UniProt AC | Q9Y4K4 |
|---|---|
| Gene Symbol | MAP4K5 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 280
- Clinical molecules 35
- Avg pChEMBL 6.9
Active Molecules (280)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KUNZDWIFPOMUOX
|
9.7 | Ki | 36 | — | |
RTYJMUXLFRYRBU
|
9.7 | Ki | 35 | — | |
UBPYILGKFZZVDX
|
9.3 | Kd | 130 | Yes | |
HKSZLNNOFSGOKW
|
9.2 | Ki | 118 | — | |
JWNPDZNEKVCWMY
|
9.2 | Kd | 57 | Yes | |
DADQIQQXJSXLAV
|
9.1 | Ki | 5 | — | |
ORRHVRJUSPCILV
|
8.9 | Ki | 16 | — | |
ZCCJKVBTHCOISJ
|
8.8 | Ki | 46 | — | |
CQBBMNXXVMOFCA
|
8.4 | Ki | 39 | — | |
DPEXRCOBPACFOO
|
8.4 | Ki | 36 | — | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
KHGPYYFCIAISBU
|
8.3 | Ki | 31 | — | |
LHQWPYOYDRVMFI
|
8.3 | Ki | 21 | — | |
XCHWBXBDZRJVDP
|
8.3 | Ki | 51 | — | |
XKZQZMSAWVDRSP
|
8.3 | Ki | 39 | Yes | |
UPJZIJDYXTYCDV
|
8.2 | Kd | 5 | — | |
VRQMAABPASPXMW
|
8.2 | Kd | 10 | — | |
NRGYZNJPCGRCLV
|
8.2 | Ki | 52 | — | |
NWAUBAGBGOPJLF
|
8.2 | Ki | 51 | Yes | |
SFPWNTQWFFNJIH
|
8.2 | Ki | 48 | — | |
ZGDSBEUMPIMXBM
|
8.2 | Ki | 42 | — | |
IFPPYSWJNWHOLQ
|
8.1 | Ki | 52 | Yes | |
LGHBDVLAHHANMX
|
8.1 | Ki | 53 | — | |
MQRDVGBWWVWMEN
|
8.1 | Ki | 47 | — | |
OOMBFNDWQIGHEK
|
8.1 | Kd | 22 | — | |
RYAVJHIPOWNWDE
|
8.1 | Ki | 38 | — | |
MFMXAWQGPQXDRJ
|
8.0 | Ki | 27 | — | |
WVUNYSQLFKLYNI
|
8.0 | Kd | 46 | Yes | |
ZBCMHWUFWQFPLV
|
8.0 | IC50 | 9 | — | |
KNACLJBHKVSTDL
|
7.9 | Ki | 40 | — | |
NFMGZVPRGVERNN
|
7.9 | Ki | 44 | — | |
SRUYMJRFVGLQDV
|
7.9 | Ki | 37 | — | |
HKZKELVPGXJIMW
|
7.8 | Ki | 41 | — | |
MTCHQDWUHQADSY
|
7.8 | Ki | 29 | — | |
WINHZLLDWRZWRT
|
7.8 | Ki | 66 | — | |
XKFTZKGMDDZMJI
|
7.8 | Ki | 56 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 213 | — | |
ACNCCUVYXQGPKZ
|
7.7 | Ki | 31 | — | |
GSXRCPJTNIGKSZ
|
7.7 | Ki | 43 | — | |
JZTOUVBEZONDKA
|
7.7 | Ki | 80 | — | |
DSSNAGYVGTYAGH
|
7.7 | IC50 | 10 | — | |
SLEWGGZPOQNVSU
|
7.6 | Kd | 22 | — | |
ADMFLILDQJSEIK
|
7.6 | Ki | 72 | — | |
ISVHLTLEHRZKJC
|
7.6 | Ki | 19 | — | |
KDLLVDABAMKMLD
|
7.6 | Ki | 4 | — | |
PTVPBWWDGZSEAF
|
7.6 | Ki | 63 | — | |
RWTXXGPUNDKBLW
|
7.6 | IC50 | 4 | — | |
RYYNGWLOYLRZLK
|
7.6 | Ki | 104 | — | |
ZKLJKKASNXVQBZ
|
7.6 | Ki | 27 | — |