Target Details
| UniProt AC | Q9Y478 |
|---|---|
| Gene Symbol | PRKAB1 |
| Protein Name | 5'-AMP-activated protein kinase subunit beta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16561 (AMPK1_CBM) PF04739 (AMPKBI) |
Summary
- Multi-target molecules 65
- Clinical molecules 5
- Avg pChEMBL 7.18
KEGG Pathways (16)
- AMPK signaling pathway
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Apelin signaling pathway
- Circadian rhythm
- FoxO signaling pathway
- Glucagon signaling pathway
- Hypertrophic cardiomyopathy
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- Non-alcoholic fatty liver disease
- Oxytocin signaling pathway
- Thermogenesis
- Tight junction
Active Molecules (65)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VCLMLPXAUIQEEM
|
6.6 | IC50 | 7 | — | |
OOQJIJYKWXLQNC
|
6.5 | IC50 | 16 | Yes | |
NDIUYMHNCUTVGE
|
6.5 | Ki | 25 | — | |
GCQRNJUDAAOEJK
|
6.4 | Kd | 3 | — | |
ZXOKHOODFVNZIC
|
6.3 | IC50 | 7 | — | |
CTESJDQKVOEUOY
|
6.3 | Kd | 3 | — | |
CQZOSLVFDRPCFJ
|
6.3 | IC50 | 7 | — | |
DXLXRNZCYAYUED
|
6.3 | IC50 | 2 | — | |
JBRGOJOHEISXNB
|
6.2 | Kd | 3 | — | |
WNLKAYDTKKISBN
|
6.2 | IC50 | 7 | — | |
INGGFDWTZNSBPY
|
6.1 | IC50 | 7 | — | |
NGDYCJGYGAYDIM
|
6.1 | IC50 | 7 | — | |
ZWIGVNWZHBPXNS
|
6.1 | IC50 | 7 | — | |
BUMYTKZYNNGHLL
|
6.0 | IC50 | 7 | — | |
XBGWAKUQSRNWMA
|
6.0 | IC50 | 4 | — |