Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QZIYOWZOZNSBGJ
|
6.8 | IC50 | 3 | — | |
UKWWUFBDIVBOBD
|
6.8 | IC50 | 5 | — | |
YCEAZZWLNZYSCL
|
6.8 | IC50 | 5 | — | |
AINKQRBPBUTJRM
|
6.7 | IC50 | 5 | — | |
PAEFKCSDRFLRMD
|
6.7 | IC50 | 5 | — | |
MGAHZVJVMCCAOO
|
6.7 | IC50 | 2 | — | |
XXIXFZAUCITSCM
|
6.7 | IC50 | 7 | — | |
AMUFSGPBIFOSNV
|
6.7 | IC50 | 3 | — | |
FXZCSYXEGFNOPO
|
6.7 | IC50 | 2 | — | |
OEVQTWCGWDOIFZ
|
6.7 | IC50 | 6 | — | |
WKYMGORXOQPTTO
|
6.7 | IC50 | 9 | — | |
ACOQCSBMVFAWQV
|
6.7 | IC50 | 8 | — | |
AKTCVLPOZVXXJU
|
6.7 | IC50 | 4 | — | |
OEVQTWCGWDOIFZ
|
6.7 | IC50 | 7 | — | |
BOSSBLQXHFNQIF
|
6.7 | IC50 | 3 | — | |
GQIHUCLIFWOITE
|
6.7 | IC50 | 4 | — | |
JGBCLJZMLUMHOO
|
6.7 | Ki | 6 | — | |
OKCYRFPVWRGQBV
|
6.7 | IC50 | 5 | — | |
OUSFTKFNBAZUKL
|
6.7 | Kd | 58 | Yes | |
QCTMVDQWYGRUJK
|
6.7 | IC50 | 9 | — | |
UMYSGMXAOXMMGG
|
6.7 | IC50 | 7 | — | |
WKDIVCXCWMVLPY
|
6.7 | IC50 | 2 | — | |
HHUOQHKKRABAQB
|
6.7 | IC50 | 5 | — | |
RWUAJNWQCLQAAA
|
6.7 | IC50 | 4 | — | |
XTJRKTBELWGSDN
|
6.7 | IC50 | 6 | — | |
ABRIIMZXUFHPCH
|
6.7 | IC50 | 5 | — | |
ZHTZVZJNJGCSJO
|
6.7 | IC50 | 7 | — | |
GCSZJMUFYOAHFY
|
6.7 | IC50 | 8 | — | |
CIEDQRFRRJHOSA
|
6.7 | IC50 | 6 | — | |
CQZSVQKINMHLBO
|
6.7 | IC50 | 4 | — | |
DSQFWMPIQBMOJL
|
6.7 | IC50 | 5 | — | |
PAHHKMMVQJCPJI
|
6.7 | IC50 | 8 | — | |
SLHUAYAGWNBZQC
|
6.7 | IC50 | 2 | — | |
TZFBRBFUNGMUNQ
|
6.7 | IC50 | 3 | — | |
WWRVEMKSOIGGCS
|
6.7 | IC50 | 5 | — | |
ZHYVMENMUIEWQH
|
6.7 | IC50 | 2 | — | |
BEILWJKGWBDPRG
|
6.7 | IC50 | 7 | — | |
CVDZJUNTQGTGHF
|
6.7 | IC50 | 4 | — | |
LDYVHYUGOBDUMZ
|
6.7 | IC50 | 6 | — | |
MCNDTHVVURYHKT
|
6.7 | IC50 | 8 | — | |
ARYGGCNDASPYNG
|
6.6 | IC50 | 3 | — | |
KBEZZFIQPRMPRG
|
6.6 | IC50 | 5 | — | |
GFSFWVNETAIFJQ
|
6.6 | IC50 | 2 | — | |
XDJCLCLBSGGNKS
|
6.6 | IC50 | 21 | — | |
BYUPNMOFJSAIHN
|
6.6 | IC50 | 6 | — | |
FGBSSPMQGRUJPS
|
6.6 | IC50 | 10 | — | |
RUQXGVGYNKIGJD
|
6.6 | IC50 | 6 | — | |
ACOQCSBMVFAWQV
|
6.6 | IC50 | 6 | — | |
CXOICQRVGSVVHC
|
6.6 | IC50 | 2 | — | |
UBUJLBVNZCRWPX
|
6.6 | IC50 | 7 | — |