Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTHYGYNOCOBONC
|
6.9 | IC50 | 4 | — | |
XZWVOUQIYLZUCJ
|
6.9 | Ki | 23 | — | |
BGVLELSCIHASRV
|
6.9 | Kd | 12 | — | |
BGVLELSCIHASRV
|
6.9 | Kd | 12 | — | |
BUDHBLBYISRDCR
|
6.9 | IC50 | 2 | — | |
CMEHUCXLRATIIB
|
6.9 | IC50 | 2 | — | |
KOMXYYABYRRJBD
|
6.9 | IC50 | 3 | — | |
MQSQPFAQNYDQLL
|
6.9 | IC50 | 5 | — | |
URXJBXVGNBGIJA
|
6.9 | IC50 | 9 | — | |
VBYRFFCBZNEHAL
|
6.9 | IC50 | 4 | — | |
YELPLVUUDHOICI
|
6.9 | IC50 | 4 | — | |
JBWDTSLHUJHODF
|
6.9 | IC50 | 8 | — | |
XTJRKTBELWGSDN
|
6.9 | IC50 | 8 | — | |
CUXJJQQRHNRQEY
|
6.9 | IC50 | 4 | — | |
OWEQZGPRBRSUEF
|
6.9 | IC50 | 2 | — | |
SIVLENRHVVVPKJ
|
6.9 | IC50 | 2 | — | |
DPSFKKBIIZTWDA
|
6.9 | IC50 | 3 | — | |
GIQDYWGEMOCDSN
|
6.9 | IC50 | 5 | — | |
JQHTYMOOIFVIJV
|
6.9 | IC50 | 5 | — | |
PINHQPCEXCQCGH
|
6.9 | IC50 | 2 | — | |
FTZQWKAIKYEWPM
|
6.8 | IC50 | 2 | — | |
RVNDFXJEYCICIV
|
6.8 | IC50 | 7 | — | |
ZUADZDBGZDSSAB
|
6.8 | IC50 | 5 | — | |
DXVSNYWBRDTHFF
|
6.8 | IC50 | 7 | — | |
IEAUISSAHDPODS
|
6.8 | IC50 | 2 | — | |
AAYFHKFUAWLHMY
|
6.8 | IC50 | 5 | — | |
VFLDPWHFBUODDF
|
6.8 | IC50 | 25 | — | |
LZTDWHFXSWDVAG
|
6.8 | IC50 | 7 | — | |
UXVJSLNUZNAQHS
|
6.8 | IC50 | 2 | — | |
YDTHCIZMSQZYMR
|
6.8 | IC50 | 9 | — | |
LRPOHOOPSDHHPW
|
6.8 | IC50 | 5 | — | |
QVYXLOYBJBMXNP
|
6.8 | IC50 | 7 | — | |
SHHUBFYLSRKFFE
|
6.8 | IC50 | 2 | — | |
CWJLAVRXVFHDSJ
|
6.8 | IC50 | 13 | — | |
DWTNLZZEPSCAIH
|
6.8 | Ki | 25 | — | |
GJOXRIYWDHESDF
|
6.8 | Ki | 27 | — | |
HHSNDNONCUTNQR
|
6.8 | IC50 | 7 | — | |
MVRRAWJPZXNFMK
|
6.8 | IC50 | 6 | — | |
OAKDCYWBXLUPQD
|
6.8 | IC50 | 4 | — | |
SYLTYCLPHHSEIJ
|
6.8 | Ki | 27 | — | |
UFGCTWUIESUHQP
|
6.8 | IC50 | 7 | — | |
UIRCQOKSJDLYBB
|
6.8 | Ki | 50 | — | |
BXNJHAXVSOCGBA
|
6.8 | IC50 | 14 | — | |
CEWIXDGUKGVYDQ
|
6.8 | IC50 | 7 | — | |
HUFHINCQVVFZJG
|
6.8 | IC50 | 2 | — | |
MFLKPCAUPXBTPC
|
6.8 | IC50 | 6 | — | |
VGWCJGBQHCMHNJ
|
6.8 | IC50 | 8 | — | |
CROVEFPUGGIVBG
|
6.8 | IC50 | 2 | — | |
BAUOZGQJLRLMNO
|
6.8 | IC50 | 4 | — | |
UTDNMHFLZJFPPY
|
6.8 | IC50 | 4 | — |