Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JANQPHRPUAYQTA
|
7.0 | IC50 | 5 | — | |
LZRHAZRGHSSHLR
|
7.0 | IC50 | 7 | — | |
BUDHVVXPBGMAPV
|
7.0 | IC50 | 11 | — | |
FKRHOHUJMCOWDZ
|
7.0 | IC50 | 5 | — | |
KAEULNCNLILYLK
|
7.0 | IC50 | 4 | — | |
NBIWQDNWQHQXFS
|
7.0 | IC50 | 5 | — | |
AQDWDWAYVBQMAM
|
7.0 | IC50 | 7 | — | |
OCVVFPATGNRPNO
|
7.0 | IC50 | 2 | — | |
QLSWEZZOYCDEGC
|
7.0 | IC50 | 5 | — | |
RWAVDFHFFDMSHX
|
7.0 | IC50 | 4 | — | |
PCIQNDJCGPAWGK
|
7.0 | IC50 | 2 | — | |
ZBKFRVXDYILXFJ
|
7.0 | IC50 | 6 | — | |
RLTCEYSNDOXWKS
|
7.0 | IC50 | 7 | — | |
XJAODSOFFLOIKC
|
7.0 | IC50 | 2 | — | |
AHJRHEGDXFFMBM
|
7.0 | Ki | 28 | — | |
ATGVCJYHNOSZEV
|
7.0 | Ki | 23 | — | |
AYALTLXRNITQHK
|
7.0 | IC50 | 2 | — | |
BGVLELSCIHASRV
|
7.0 | Kd | 11 | — | |
DFCORNPUKFIPDM
|
7.0 | IC50 | 2 | — | |
DPIAIAIQEINUNP
|
7.0 | IC50 | 4 | — | |
FISNDZKRNXBCLC
|
7.0 | Ki | 6 | — | |
FPFBUUBVECCCFK
|
7.0 | IC50 | 2 | — | |
JUQUOEZMUSCAFN
|
7.0 | IC50 | 3 | — | |
NJETXHOGHMMTEB
|
7.0 | IC50 | 4 | — | |
VWACUNWBMWWMPJ
|
7.0 | Ki | 18 | — | |
ZQZULRTVXPNQNP
|
7.0 | IC50 | 4 | — | |
QNWARURWFRZNNO
|
7.0 | IC50 | 7 | — | |
YGVKOSRPXIWQPQ
|
7.0 | IC50 | 4 | — | |
COYCDCAUDJBGOV
|
7.0 | IC50 | 6 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
LZUJDIWVWSRLRQ
|
7.0 | IC50 | 4 | — | |
LZUJDIWVWSRLRQ
|
7.0 | IC50 | 4 | — | |
PRJNNPMIUGYOST
|
7.0 | IC50 | 14 | — | |
SZOYOCHRMSEEMG
|
7.0 | IC50 | 7 | — | |
SZOYOCHRMSEEMG
|
7.0 | IC50 | 3 | — | |
DJHMDVUOYUYLOJ
|
7.0 | IC50 | 9 | — | |
OKBNCPDNYVDCTG
|
7.0 | IC50 | 5 | — | |
YMIDGKZVYFXIBW
|
7.0 | IC50 | 8 | — | |
AMBKAVGTUWUVBS
|
6.9 | IC50 | 8 | — | |
BULHRWBHKAVJMT
|
6.9 | IC50 | 8 | — | |
CBTNARFZVOPLBO
|
6.9 | IC50 | 8 | — | |
XDVWHWQSQJFRPP
|
6.9 | IC50 | 4 | — | |
FVIUKIZPDJZQKD
|
6.9 | IC50 | 5 | — | |
MYLYCZDLVLCRLU
|
6.9 | IC50 | 5 | — | |
CXJCGSPAPOTTSF
|
6.9 | IC50 | 6 | — | |
GHQYHWMWJLSKRP
|
6.9 | IC50 | 9 | — | |
JXQZHHAAJMQJKU
|
6.9 | IC50 | 9 | — | |
BIIVYFLTOXDAOV
|
6.9 | Ki | 31 | — | |
IEFFSHLHNYVSEF
|
6.9 | IC50 | 8 | — | |
MQJVDVMWBFSFHI
|
6.9 | IC50 | 5 | — |