Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FFESRGFMLQEDRD
|
7.2 | IC50 | 5 | — | |
NSDQDNNJFIKBKR
|
7.2 | IC50 | 6 | — | |
OJSLNTSFMXRUEG
|
7.2 | IC50 | 2 | — | |
QCHDHJOEPUQALZ
|
7.2 | IC50 | 9 | — | |
CIGFCAJNHRIRIV
|
7.2 | IC50 | 2 | — | |
HAFFBDGNUZMNIJ
|
7.2 | IC50 | 7 | — | |
HBBPDNLIBIZZFL
|
7.2 | IC50 | 7 | — | |
LMXLOYKFDZEHCS
|
7.2 | IC50 | 7 | — | |
WNKQZLFWZLQFOH
|
7.2 | IC50 | 3 | — | |
IDOKKOQIQLHASZ
|
7.2 | IC50 | 8 | — | |
BWNXEFDIXGZHPQ
|
7.1 | IC50 | 4 | — | |
FBURYRMHEHTVED
|
7.1 | IC50 | 9 | — | |
FUSZCAJFRIHBLV
|
7.1 | IC50 | 4 | — | |
JNTIINGGIOJIMW
|
7.1 | IC50 | 4 | — | |
LXDHFJUOCGKVAV
|
7.1 | IC50 | 5 | — | |
QXMXIHBLICGPMG
|
7.1 | IC50 | 9 | — | |
WQYUNADCLFWKGN
|
7.1 | IC50 | 7 | — | |
ZBYBDKHFLSHGBP
|
7.1 | IC50 | 4 | — | |
ZBYBDKHFLSHGBP
|
7.1 | IC50 | 4 | — | |
ZSZSXTFUWZNVBW
|
7.1 | IC50 | 2 | — | |
JXQZHHAAJMQJKU
|
7.1 | IC50 | 6 | — | |
FSICBNKCBMOCOY
|
7.1 | IC50 | 2 | — | |
RILDWXOQLWEXDG
|
7.1 | IC50 | 6 | — | |
VOXHNNQHNDOGSK
|
7.1 | IC50 | 4 | — | |
FTGAOPZDJRWUTG
|
7.1 | IC50 | 6 | — | |
PCUWPDUAQBAWHT
|
7.1 | IC50 | 4 | — | |
SQWZFLMPDUSYGV
|
7.1 | IC50 | 11 | — | |
SQWZFLMPDUSYGV
|
7.1 | IC50 | 8 | — | |
WLKJMISWXHORCR
|
7.1 | IC50 | 11 | — | |
YRFAWSIUIFNVQA
|
7.1 | IC50 | 9 | — | |
ZGDYBJXDIXVTLV
|
7.1 | Ki | 54 | — | |
ANKYADWZYKSCAJ
|
7.1 | IC50 | 7 | — | |
MFLKPCAUPXBTPC
|
7.1 | IC50 | 5 | — | |
NENJFZKQHYXRDQ
|
7.1 | Kd | 8 | — | |
QVLJVHWQAKYGQI
|
7.1 | IC50 | 8 | — | |
WFOMWAYINPJPDX
|
7.1 | IC50 | 9 | — | |
BIIVYFLTOXDAOV
|
7.1 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
7.1 | Kd | 82 | Yes | |
BKIAHCJPMJSHSQ
|
7.1 | IC50 | 6 | — | |
OSWHZHVVVZAPRN
|
7.1 | IC50 | 6 | — | |
UDBMFFIMVBBFKP
|
7.1 | IC50 | 3 | — | |
DYABBQVRJKEHMB
|
7.1 | IC50 | 2 | — | |
PPZINUUIYSVIGC
|
7.1 | IC50 | 6 | — | |
QJVXFDORJYYPAW
|
7.1 | IC50 | 4 | — | |
BZNZVNQDMRWLSV
|
7.1 | IC50 | 2 | — | |
GCUNCFYJKLSBKK
|
7.1 | IC50 | 5 | — | |
PMDAVRLCSZSLRH
|
7.1 | IC50 | 13 | — | |
RGKOSKZCLZXDJI
|
7.1 | IC50 | 4 | — | |
RPGZQOOZHIEPJW
|
7.1 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.1 | Kd | 18 | — |