Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KQCIEIGKPXQRLM
|
7.4 | IC50 | 6 | — | |
USYASDQVUTWEQM
|
7.4 | IC50 | 9 | — | |
OAUMCWJJYNUCIM
|
7.4 | IC50 | 5 | — | |
WAJNOEPHTZIWTO
|
7.4 | IC50 | 6 | — | |
XVVPNHZWUXCHJE
|
7.4 | IC50 | 3 | — | |
YYSXUOHHBBMQMJ
|
7.4 | IC50 | 7 | — | |
FIVWKNZKXNNFCW
|
7.4 | IC50 | 8 | — | |
VJSOYRZFTRFBFM
|
7.4 | IC50 | 5 | — | |
VZGXJTZKPDEJGJ
|
7.4 | IC50 | 2 | — | |
PEICIAVUWSXRGP
|
7.4 | IC50 | 7 | — | |
SJWUVVGOTOMGOH
|
7.4 | IC50 | 10 | — | |
VPLSDHGYIYFKRM
|
7.4 | IC50 | 2 | — | |
XTJRKTBELWGSDN
|
7.3 | IC50 | 8 | — | |
BBCSUMURJUYILA
|
7.3 | IC50 | 9 | — | |
RUQXGVGYNKIGJD
|
7.3 | IC50 | 9 | — | |
TUIPZIRQUAZXFN
|
7.3 | IC50 | 2 | — | |
BWORFRWIDWQHPL
|
7.3 | IC50 | 7 | — | |
BYMPGMQLSBLSIU
|
7.3 | IC50 | 5 | — | |
FRILKPCZRSAZON
|
7.3 | IC50 | 2 | — | |
MXEZQEFCKXVMFN
|
7.3 | IC50 | 5 | — | |
BBZSEXSOPOXLIQ
|
7.3 | Ki | 8 | — | |
GKODJBVKKLQMEY
|
7.3 | Ki | 10 | — | |
AOGIFFVMTGMFBP
|
7.3 | IC50 | 8 | — | |
GPMRASYSIQENIJ
|
7.3 | IC50 | 3 | — | |
KAGWQDFFFLWBFD
|
7.3 | IC50 | 8 | — | |
ITOTZLBIDAOTGK
|
7.3 | IC50 | 4 | — | |
ITOTZLBIDAOTGK
|
7.3 | IC50 | 4 | — | |
OHARPIGKJAKOCM
|
7.3 | IC50 | 8 | — | |
INAVVYMHODCJNF
|
7.3 | IC50 | 5 | — | |
KOEMSQCYTSQEEQ
|
7.3 | IC50 | 2 | — | |
MNPDDWGYJIGNTR
|
7.3 | IC50 | 2 | — | |
GVQSROMOXGBVJP
|
7.2 | IC50 | 2 | — | |
IFLBFWBMAWIBBZ
|
7.2 | Kd | 7 | — | |
RLTCEYSNDOXWKS
|
7.2 | IC50 | 9 | — | |
ANKYADWZYKSCAJ
|
7.2 | IC50 | 7 | — | |
QTRZNDLLYHSJSH
|
7.2 | IC50 | 9 | — | |
PAEKWZJLZMSTLB
|
7.2 | IC50 | 6 | — | |
DXVSNYWBRDTHFF
|
7.2 | IC50 | 9 | — | |
LGCHSPYDLIKTIC
|
7.2 | IC50 | 6 | — | |
PGPHHJBZEGSUNE
|
7.2 | IC50 | 21 | — | |
PGPHHJBZEGSUNE
|
7.2 | IC50 | 17 | — | |
RYWACTNAXCMTTN
|
7.2 | IC50 | 9 | — | |
UUXDJIVNVOOKFQ
|
7.2 | IC50 | 9 | — | |
AEYLJTAIDDIOBA
|
7.2 | Ki | 53 | — | |
NNPWUWSWEGWPMQ
|
7.2 | IC50 | 8 | — | |
PGPHHJBZEGSUNE
|
7.2 | IC50 | 4 | — | |
VQAZMVUNBILJGW
|
7.2 | IC50 | 5 | — | |
KCTCLVINURCCIL
|
7.2 | IC50 | 7 | — | |
UMWJBFSPIYCGRG
|
7.2 | IC50 | 7 | — | |
CQKBSRPVZZLCJE
|
7.2 | IC50 | 2 | — |