Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDSQMAISOKRJPN
|
7.6 | IC50 | 2 | — | |
WREJZZXSNOJGIW
|
7.6 | IC50 | 9 | — | |
CZWJLLBPWLUINU
|
7.6 | IC50 | 10 | — | |
WHPORTUXBLFUPA
|
7.6 | IC50 | 8 | — | |
YSODDCRKIDDXKM
|
7.6 | IC50 | 9 | — | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
OQSBQXVIMQMCES
|
7.5 | IC50 | 9 | — | |
UHOPJKMQVDXYAV
|
7.5 | IC50 | 8 | — | |
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
IJFKKIMDRSZOOW
|
7.5 | IC50 | 8 | — | |
BDWKOEXYKJGIMA
|
7.5 | IC50 | 2 | — | |
DNJISDHVBHLOGY
|
7.5 | IC50 | 2 | — | |
GEJSQZULGDKBQV
|
7.5 | IC50 | 8 | — | |
MQRHLOPPMRFMKM
|
7.5 | IC50 | 9 | — | |
SJWUVVGOTOMGOH
|
7.5 | IC50 | 12 | — | |
SJYQOVMGZOATNK
|
7.5 | IC50 | 9 | — | |
YGVLUDLFNRZMNT
|
7.5 | IC50 | 8 | — | |
ATXGVVQAUKKFAN
|
7.5 | IC50 | 4 | — | |
GDFYUGGDTISZFA
|
7.5 | IC50 | 2 | — | |
OWDVXJJCVWTPPW
|
7.5 | IC50 | 8 | — | |
PHWHNHYZZNJPLB
|
7.5 | Ki | 16 | — | |
UOVCGJXDGOGOCZ
|
7.5 | Ki | 59 | — | |
WEQRXDXDFLBIDK
|
7.5 | IC50 | 8 | — | |
WFOMWAYINPJPDX
|
7.5 | IC50 | 9 | — | |
CHQYAWLKOUOTQO
|
7.5 | IC50 | 7 | — | |
HJEKFRDOAYXXRU
|
7.5 | IC50 | 8 | — | |
IJFKKIMDRSZOOW
|
7.5 | IC50 | 9 | — | |
OAAPSDVPLURZJC
|
7.5 | IC50 | 2 | — | |
UVJQEKJPAVSBTA
|
7.5 | IC50 | 8 | — | |
KRXQWLCJHMDEDM
|
7.5 | IC50 | 8 | — | |
XGDCSHCKBNJGMN
|
7.5 | IC50 | 2 | — | |
YHZQZEGQCKWCLP
|
7.5 | IC50 | 9 | — | |
IMSFHJBONZQKCR
|
7.4 | IC50 | 2 | — | |
DSCUTYQYWCTFQL
|
7.4 | IC50 | 6 | — | |
MDPBVLVUPMAUIA
|
7.4 | IC50 | 2 | — | |
ZDINVWCJHPMIKS
|
7.4 | IC50 | 2 | — | |
FEZCHKAGMYXVNX
|
7.4 | IC50 | 6 | — | |
LQLBWZJHRARWDB
|
7.4 | IC50 | 6 | — | |
PVFNDFZQGWYILU
|
7.4 | IC50 | 3 | — | |
RMQRHTAARSAOHF
|
7.4 | IC50 | 5 | — | |
YGXHQYJKJUFSJI
|
7.4 | IC50 | 14 | — | |
TYVKILZNVZGMIM
|
7.4 | IC50 | 2 | — | |
BQYDGSNDLAZAEW
|
7.4 | Ki | 13 | — | |
DCHAEDURAZJASA
|
7.4 | IC50 | 9 | — | |
JLTBOCSFMNSLFH
|
7.4 | Ki | 9 | — | |
OSVUGUHRKMMBSE
|
7.4 | Kd | 170 | — | |
RQFGUPSBOAVFSQ
|
7.4 | IC50 | 2 | — | |
SOHWYEVCBPDAIO
|
7.4 | IC50 | 3 | — | |
YSBCFQVEEKUZSU
|
7.4 | IC50 | 7 | — | |
JGJABYQWCCWLPP
|
7.4 | IC50 | 4 | — |