Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HXESDBWWDYJEJQ
|
7.9 | Ki | 10 | — | |
VCCCOYOXNKTQFO
|
7.9 | IC50 | 9 | — | |
MLAPBLMPGXKRBF
|
7.9 | IC50 | 3 | — | |
ROPFCXUWNMYMSW
|
7.9 | IC50 | 10 | — | |
UTGHIUITNUXCRZ
|
7.9 | IC50 | 2 | — | |
PTTXGLLPYLIZCU
|
7.9 | IC50 | 2 | — | |
DCJOTKUJWJFCSP
|
7.8 | IC50 | 9 | — | |
OYDWEMSWMQKSLK
|
7.8 | IC50 | 8 | — | |
YAXGFAAKCUOWNM
|
7.8 | IC50 | 9 | — | |
OVVHFDIQCYTOAS
|
7.8 | IC50 | 9 | — | |
RAQBQAXSLHDSKW
|
7.8 | IC50 | 8 | — | |
UUIPRATXTHJYHH
|
7.8 | IC50 | 3 | — | |
CRKQBJZCCHKEGI
|
7.8 | Ki | 20 | — | |
RGNHKJWHFIPHIM
|
7.8 | Ki | 66 | — | |
RRAMBEGOYIJQHY
|
7.8 | Ki | 11 | — | |
WDARYLSSWBWVCU
|
7.8 | Ki | 49 | — | |
ZGZVRPRSFXRGCF
|
7.8 | Ki | 76 | — | |
JJUHKRNDDMOYGK
|
7.8 | IC50 | 3 | — | |
UTGHIUITNUXCRZ
|
7.8 | IC50 | 2 | — | |
VAXXXDBEUYQWBN
|
7.8 | IC50 | 2 | — | |
ZYVXTMKTGDARKR
|
7.8 | IC50 | 6 | — | |
GHNZOLKSIZOQCZ
|
7.8 | IC50 | 2 | — | |
SJWUVVGOTOMGOH
|
7.8 | IC50 | 9 | — | |
YJKPCYDSZXIODK
|
7.8 | IC50 | 8 | — | |
CIJWGWNHXQYIJC
|
7.7 | IC50 | 5 | — | |
KNLSVEADBVICIJ
|
7.7 | IC50 | 5 | — | |
LUKGZXVCOQQBHB
|
7.7 | IC50 | 2 | — | |
QDNBLKZVYODRLC
|
7.7 | IC50 | 5 | — | |
SDAAXACYZBWYTQ
|
7.7 | IC50 | 2 | — | |
YBASBPWQGVPOIX
|
7.7 | IC50 | 2 | — | |
ZLFXEVGPZWFVCB
|
7.7 | IC50 | 2 | — | |
JBWDTSLHUJHODF
|
7.7 | IC50 | 9 | — | |
WYEVMOFRKALLJA
|
7.7 | IC50 | 4 | — | |
YHZQZEGQCKWCLP
|
7.7 | IC50 | 9 | — | |
JUSBGYZKUCMHQQ
|
7.7 | IC50 | 2 | — | |
CGRDYMCBGXJNLR
|
7.7 | IC50 | 9 | — | |
JHKYWRMDSIQKSV
|
7.7 | IC50 | 2 | — | |
WHPORTUXBLFUPA
|
7.7 | IC50 | 9 | — | |
MOYYMSNZEWQWQJ
|
7.7 | IC50 | 3 | — | |
AKNIGLLNHUTMPO
|
7.6 | IC50 | 9 | — | |
JBWDTSLHUJHODF
|
7.6 | IC50 | 9 | — | |
PBVAHEBIEXXNNA
|
7.6 | IC50 | 4 | — | |
QTRZNDLLYHSJSH
|
7.6 | IC50 | 9 | — | |
GRHRWVRWLAIBGN
|
7.6 | IC50 | 5 | — | |
VRGNMDTYOWQXQC
|
7.6 | IC50 | 8 | — | |
VRGNMDTYOWQXQC
|
7.6 | IC50 | 5 | — | |
WREJZZXSNOJGIW
|
7.6 | IC50 | 8 | — | |
HZPACYSNLOCDLW
|
7.6 | Ki | 48 | — | |
NFPDLDFOSLPKHQ
|
7.6 | IC50 | 2 | — | |
XUFLBSMTYMFOQH
|
7.6 | Ki | 43 | — |