Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVQOYBIBWBAHKH
|
8.3 | IC50 | 12 | — | |
HFJRGZBUEXFBMO
|
8.2 | IC50 | 2 | — | |
BNPUEXLGIHXXJP
|
8.2 | IC50 | 2 | — | |
CIICGXXZCWRFQE
|
8.2 | IC50 | 7 | — | |
IVSYLIPATGYBCZ
|
8.2 | IC50 | 7 | — | |
UGYUFJPHSWYELP
|
8.2 | IC50 | 8 | — | |
YSBCFQVEEKUZSU
|
8.2 | IC50 | 9 | — | |
MUOKSQABCJCOPU
|
8.2 | IC50 | 36 | — | |
UZWDCWONPYILKI
|
8.2 | IC50 | 47 | — | |
ZBELDPMWYXDLNY
|
8.2 | IC50 | 4 | — | |
GXCOUFPTCZUTEE
|
8.2 | IC50 | 10 | — | |
FFJGYBJUQCZAAY
|
8.2 | IC50 | 5 | — | |
MGEGGAFJSKMJJD
|
8.2 | IC50 | 5 | — | |
PVMYRLVGSWLCSL
|
8.2 | IC50 | 2 | — | |
VFLPOFHPMNYCOH
|
8.2 | IC50 | 7 | — | |
XCTYEZWILVGTGO
|
8.2 | IC50 | 9 | — | |
CHQYAWLKOUOTQO
|
8.1 | IC50 | 20 | — | |
QCJWUXFCDRVWGH
|
8.1 | IC50 | 2 | — | |
QTRQYFCAAHDIDR
|
8.1 | IC50 | 2 | — | |
UZIATSFXNVOVFE
|
8.1 | IC50 | 9 | — | |
ZGFYGZLBXCHRCV
|
8.1 | IC50 | 2 | — | |
CLEGDJQQHUTCOW
|
8.1 | Ki | 43 | — | |
JCJWCXBSDFGDSJ
|
8.1 | IC50 | 3 | — | |
KBMQGIPVJGXLOU
|
8.1 | IC50 | 7 | — | |
MRWURALZVKJHPD
|
8.1 | IC50 | 2 | — | |
SBYPANVVFZBWDF
|
8.1 | IC50 | 9 | — | |
YORVMWUGDVGXOQ
|
8.1 | IC50 | 8 | — | |
DXVSNYWBRDTHFF
|
8.1 | IC50 | 10 | — | |
FIVWKNZKXNNFCW
|
8.1 | IC50 | 9 | — | |
FWFWXUJORMCFKY
|
8.1 | IC50 | 3 | — | |
JAJFJEDUYYFVEE
|
8.1 | IC50 | 2 | — | |
KSIRCFGDZWDBAM
|
8.1 | IC50 | 2 | — | |
SKKBUBMBPCJYKW
|
8.1 | IC50 | 9 | — | |
KIMRTWGQATWAQF
|
8.0 | IC50 | 2 | — | |
ANBPRTXIECGGEM
|
8.0 | IC50 | 2 | — | |
CEFPPDKMUCDGCU
|
8.0 | IC50 | 3 | — | |
DKXHSOUZPMHNIZ
|
8.0 | Ki | 51 | Yes | |
HAPIHWIYVZOFQR
|
8.0 | IC50 | 4 | — | |
JFDRONLMXPRQPP
|
8.0 | IC50 | 9 | — | |
KHQYSWUSDRSLMP
|
8.0 | IC50 | 2 | — | |
ORBNLRQBHQLUIW
|
8.0 | IC50 | 2 | — | |
WCGVAQKYQAEAIH
|
8.0 | IC50 | 2 | — | |
YNGHSMIWDSRNCH
|
8.0 | IC50 | 2 | — | |
JMENQRYRZLNDDO
|
8.0 | IC50 | 2 | — | |
KUFCYNGJQRKYSQ
|
8.0 | IC50 | 2 | — | |
SLKHMZQUNIHINK
|
8.0 | IC50 | 10 | — | |
CLIWAKTWXZNUAC
|
8.0 | IC50 | 2 | — | |
BWKADHBOXYDZFU
|
7.9 | IC50 | 10 | — | |
OGPJOAYIAOEJAM
|
7.9 | IC50 | 8 | — | |
PPALZSWDMRGSQV
|
7.9 | IC50 | 5 | — |