Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AQLWSCZCZJWUMZ
|
6.6 | IC50 | 6 | — | |
BLQYVHBZHAISJM
|
6.6 | Ki | 54 | — | |
DYHKEGKDOOZETF
|
6.6 | IC50 | 9 | — | |
JRNJNYBQQYBCLE
|
6.6 | Kd | 40 | Yes | |
KZHOWDULHMQJNY
|
6.6 | IC50 | 2 | — | |
MYHMILRQDXANLR
|
6.6 | IC50 | 2 | — | |
QNLMLEYLZSGBHP
|
6.6 | Ki | 8 | — | |
RFVBRKXQYUDGIO
|
6.6 | Ki | 23 | — | |
UBPOBEKAVPQZHZ
|
6.6 | IC50 | 5 | — | |
YDTHCIZMSQZYMR
|
6.6 | IC50 | 7 | — | |
DGSCWEKDRWDCOB
|
6.6 | IC50 | 5 | — | |
KJFGBDYZIORKKA
|
6.6 | IC50 | 2 | — | |
PCHKPVIQAHNQLW
|
6.6 | IC50 | 8 | — | |
LKROTCXRJRCMTD
|
6.6 | IC50 | 4 | — | |
YVSLJAICTSVCDB
|
6.6 | IC50 | 6 | — | |
KQZBWTMAFLOSPA
|
6.6 | IC50 | 8 | — | |
LASLZTNNTZVYMJ
|
6.6 | IC50 | 4 | — | |
MPXAWSABMVLIBU
|
6.6 | IC50 | 6 | — | |
UGUVGLVHRPLWRS
|
6.6 | IC50 | 3 | — | |
UGUVGLVHRPLWRS
|
6.6 | IC50 | 3 | — | |
CRLFBJGERQILPV
|
6.6 | Ki | 2 | — | |
QTRZNDLLYHSJSH
|
6.6 | IC50 | 7 | — | |
JOCUCEXJBMSIMH
|
6.5 | IC50 | 2 | — | |
OVPNQJVDAFNBDN
|
6.5 | Kd | 44 | Yes | |
IXTKPNOXAVTBCW
|
6.5 | IC50 | 4 | — | |
TWKWEBMGDALHPN
|
6.5 | IC50 | 9 | — | |
YORVMWUGDVGXOQ
|
6.5 | IC50 | 8 | — | |
KCTCLVINURCCIL
|
6.5 | IC50 | 6 | — | |
KKVKVCZEAYHBCN
|
6.5 | IC50 | 2 | — | |
MHURZKJMJCNXDR
|
6.5 | IC50 | 5 | — | |
QASZHVBKEAXRMM
|
6.5 | IC50 | 3 | — | |
WCJBJECTLLTBHS
|
6.5 | IC50 | 2 | — | |
ABMAOGVUUQCYHD
|
6.5 | IC50 | 2 | — | |
DYIOAOFYWZXKEX
|
6.5 | IC50 | 4 | — | |
DYIOAOFYWZXKEX
|
6.5 | IC50 | 4 | — | |
GWXPHWSUMLUDPO
|
6.5 | Ki | 11 | — | |
HOLVNBCAYHKGJL
|
6.5 | IC50 | 5 | — | |
JFKIXRTUZAZONT
|
6.5 | Ki | 6 | — | |
KDJGCVHPUMHUOL
|
6.5 | Ki | 11 | — | |
OUJZYQBEFNDJQN
|
6.5 | Ki | 71 | — | |
OWRXHGAFWZFFCW
|
6.5 | Ki | 113 | — | |
PIMQWRZWLQKKBJ
|
6.5 | Ki | 5 | — | |
XOBINHQHMGZFDI
|
6.5 | IC50 | 5 | — | |
FRPGBGWSLAGPND
|
6.5 | IC50 | 7 | — | |
XXTRJPVJIAZBBR
|
6.5 | IC50 | 2 | — | |
BIDTZRBRWDXWHU
|
6.5 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 91 | Yes | |
HFLXYSRIPKXGOQ
|
6.5 | IC50 | 4 | — | |
HVEXJKQESNIDLM
|
6.5 | Kd | 10 | — |